XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa MAP2K6
DVkPSNVLINALGQVK
Lys2
2.1
10
uM
XMD8-92 PC-3 MAP2K6
DVkPSNVLINALGQVK
Lys2
7.2
10
uM
XMD8-92 PC-3 MAP2K6
HVPSGQIMAVkR
Lys1
1.8
10
uM
XMD8-92 HeLa MAP3K1
DVkGANLLIDSTGQR
Lys2
-33.3
10
uM
XMD8-92 PC-3 M3K2
ELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
24.4
10
uM
XMD8-92 HeLa M3K2,MAP3K3
DIkGANILR
Lys2
-1.6
10
uM
XMD8-92 PC-3 M3K2,MAP3K3
DIkGANILR
Lys2
0.4
10
uM
XMD8-92 HeLa MAP3K4
DIkGANIFLTSSGLIK
Lys2
-5.9
10
uM
XMD8-92 PC-3 MAP3K4
DIkGANIFLTSSGLIK
Lys2
10.6
10
uM
XMD8-92 HeLa MAP3K5,MAP3K6,MAP3K7
IAIkEIPERDSR
Lys1
3.2
10
uM
XMD8-92 HeLa MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
3.8
10
uM
XMD8-92 PC-3 MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
4.0
10
uM
XMD8-92 HeLa MAST2,MAST4
DLkPDNLLVTSMGHIK
Lys2
9.1
10
uM
XMD8-92 HeLa MAST3
DLkPDNLLITSLGHIK
Lys2
9.2
10
uM
XMD8-92 PC-3 MAST3
DLkPDNLLITSLGHIK
Lys2
7.9
10
uM
XMD8-92 HeLa MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
-11.4
10
uM
XMD8-92 PC-3 MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
15.6
10
uM
XMD8-92 HeLa MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
18.1
10
uM
XMD8-92 PC-3 MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
12.5
10
uM
XMD8-92 HeLa MSK1,MSK2_domain1
VLGTGAYGkVFLVR
ATP Loop
-4.9
10
uM
XMD8-92 HeLa MSK1_domain1
DIkLENILLDSNGHVVLTDFGLSK
Lys2
-48.1
10
uM
XMD8-92 HeLa MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
-4.1
10
uM
XMD8-92 PC-3 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
1.3
10
uM
XMD8-92 PC-3 MST1,MST2
DIkAGNILLNTEGHAK
Lys2
-9.4
10
uM
XMD8-92 HeLa MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
13.6
10
uM