XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-92 | HeLa | MAP2K6 | DVkPSNVLINALGQVK | Lys2 | 2.1 | 10 | uM |
XMD8-92 | PC-3 | MAP2K6 | DVkPSNVLINALGQVK | Lys2 | 7.2 | 10 | uM |
XMD8-92 | PC-3 | MAP2K6 | HVPSGQIMAVkR | Lys1 | 1.8 | 10 | uM |
XMD8-92 | HeLa | MAP3K1 | DVkGANLLIDSTGQR | Lys2 | -33.3 | 10 | uM |
XMD8-92 | PC-3 | M3K2 | ELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | 24.4 | 10 | uM |
XMD8-92 | HeLa | M3K2,MAP3K3 | DIkGANILR | Lys2 | -1.6 | 10 | uM |
XMD8-92 | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | 0.4 | 10 | uM |
XMD8-92 | HeLa | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | -5.9 | 10 | uM |
XMD8-92 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | 10.6 | 10 | uM |
XMD8-92 | HeLa | MAP3K5,MAP3K6,MAP3K7 | IAIkEIPERDSR | Lys1 | 3.2 | 10 | uM |
XMD8-92 | HeLa | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 3.8 | 10 | uM |
XMD8-92 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 4.0 | 10 | uM |
XMD8-92 | HeLa | MAST2,MAST4 | DLkPDNLLVTSMGHIK | Lys2 | 9.1 | 10 | uM |
XMD8-92 | HeLa | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 9.2 | 10 | uM |
XMD8-92 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 7.9 | 10 | uM |
XMD8-92 | HeLa | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | -11.4 | 10 | uM |
XMD8-92 | PC-3 | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | 15.6 | 10 | uM |
XMD8-92 | HeLa | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 18.1 | 10 | uM |
XMD8-92 | PC-3 | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 12.5 | 10 | uM |
XMD8-92 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | -4.9 | 10 | uM |
XMD8-92 | HeLa | MSK1_domain1 | DIkLENILLDSNGHVVLTDFGLSK | Lys2 | -48.1 | 10 | uM |
XMD8-92 | HeLa | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | -4.1 | 10 | uM |
XMD8-92 | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 1.3 | 10 | uM |
XMD8-92 | PC-3 | MST1,MST2 | DIkAGNILLNTEGHAK | Lys2 | -9.4 | 10 | uM |
XMD8-92 | HeLa | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 13.6 | 10 | uM |