XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-92 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | -4.9 | 10 | uM |
| XMD8-92 | PC-3 | ILK | WQGNDIVVkVLK | Lys1 | 17.7 | 10 | uM |
| XMD8-92 | PC-3 | IRAK1 | AIQFLHQDSPSLIHGDIkSSNVLLDER | Lys2 | 4.3 | 10 | uM |
| XMD8-92 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | 2.8 | 10 | uM |
| XMD8-92 | PC-3 | IRAK4 | DIkSANILLDEAFTAK | Lys2 | 2.8 | 10 | uM |
| XMD8-92 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | -10.9 | 10 | uM |
| XMD8-92 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | -10.4 | 10 | uM |
| XMD8-92 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | -18.1 | 10 | uM |
| XMD8-92 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | 6.5 | 10 | uM |
| XMD8-92 | HeLa | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | -0.1 | 10 | uM |
| XMD8-92 | PC-3 | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | 10.6 | 10 | uM |
| XMD8-92 | PC-3 | KHS1 | NVHTGELAAVkIIK | Lys1 | -7.6 | 10 | uM |
| XMD8-92 | HeLa | LATS1 | ALYATkTLR | Lys1 | 0.4 | 10 | uM |
| XMD8-92 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -8.3 | 10 | uM |
| XMD8-92 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | 7.3 | 10 | uM |
| XMD8-92 | HeLa | LOK | DLkAGNVLMTLEGDIR | Lys2 | 15.0 | 10 | uM |
| XMD8-92 | PC-3 | LOK | DLkAGNVLMTLEGDIR | Lys2 | 7.0 | 10 | uM |
| XMD8-92 | HeLa | LOK | NKETGALAAAkVIETK | Lys1 | -9.7 | 10 | uM |
| XMD8-92 | PC-3 | LOK | NKETGALAAAkVIETK | Lys1 | 4.0 | 10 | uM |
| XMD8-92 | HeLa | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | -11.6 | 10 | uM |
| XMD8-92 | PC-3 | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | 0.0 | 10 | uM |
| XMD8-92 | HeLa | MAP2K3 | DVkPSNVLINK | Lys2 | 8.3 | 10 | uM |
| XMD8-92 | PC-3 | MAP2K3 | DVkPSNVLINK | Lys2 | 1.5 | 10 | uM |
| XMD8-92 | PC-3 | MAP2K4 | MVHKPSGQIMAVkR | Lys1 | 6.9 | 10 | uM |
| XMD8-92 | PC-3 | MAP2K4 | DIkPSNILLDR | Lys2 | 2.2 | 10 | uM |