XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD8-85 | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | -10.1 | 10 | uM |
XMD8-85 | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | -34.8 | 10 | uM |
XMD8-85 | HeLa | KSR1,KSR2 | SkNVFYDNGK | Protein Kinase Domain | -0.8 | 10 | uM |
XMD8-85 | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | -13.5 | 10 | uM |
XMD8-85 | HeLa | LYN | VAVkTLKPGTMSVQAFLEEANLMK | Lys1 | -34.8 | 10 | uM |
XMD8-85 | PC-3 | M3K2 | VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -45.7 | 10 | uM |
XMD8-85 | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | -12.2 | 10 | uM |
XMD8-85 | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | -15.8 | 10 | uM |
XMD8-85 | PC-3 | MARK2 | EVAVkIIDKTQLNSSSLQK | Lys1 | -3.9 | 10 | uM |
XMD8-85 | PC-3 | MARK3,MARK4 | EVAIkIIDK | Lys1 | -5.9 | 10 | uM |
XMD8-85 | HeLa | MASTL | LYAVkVVK | Lys1 | -12.0 | 10 | uM |
XMD8-85 | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | 15.3 | 10 | uM |
XMD8-85 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | 16.7 | 10 | uM |
XMD8-85 | HeLa | p38a | DLkPSNLAVNEDCELK | Lys2 | -25.7 | 10 | uM |
XMD8-85 | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | -25.7 | 10 | uM |
XMD8-85 | HeLa | MK14 | QELNkTIWEVPER | Other | -19.8 | 10 | uM |
XMD8-85 | PC-3 | MK14 | QELNkTIWEVPER | Other | -2.9 | 10 | uM |
XMD8-85 | HeLa | PAN3 | VMDPTkILITGK | -7.7 | 10 | uM | |
XMD8-85 | HeLa | PEK | DLkPSNIFFTMDDVVK | Lys2 | -32.9 | 10 | uM |
XMD8-85 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 9.3 | 10 | uM |
XMD8-85 | HeLa | PIK3CG | KkPLWLEFK | ATP | -13.4 | 10 | uM |
XMD8-85 | HeLa | PKN1 | GHFGkVLLSEFRPSGELFAIK | Lys1 | -20.5 | 10 | uM |
XMD8-85 | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | 2.6 | 10 | uM |
XMD8-85 | PC-3 | ROCK1 | kLQLELNQER | Other | -11.7 | 10 | uM |
XMD8-85 | PC-3 | RON | IQCAIkSLSR | Lys1 | -0.5 | 10 | uM |