XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
-25.3
10
uM
XMD8-85 PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
9.6
10
uM
XMD8-85 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
31.1
10
uM
XMD8-85 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
-26.7
10
uM
XMD8-85 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-3.5
10
uM
XMD8-85 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
13.1
10
uM
XMD8-85 PC-3 TLK2
YVAVkIHQLNK
Lys1
5.0
10
uM
XMD8-85 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-14.6
10
uM
XMD8-85 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-17.8
10
uM
XMD8-85 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-7.8
10
uM
XMD8-85 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
-6.3
10
uM
XMD8-85 HeLa MLTK
WISQDKEVAVKk
Lys1
-11.5
10
uM
XMD8-85 PC-3 MLTK
WISQDKEVAVKk
Lys1
0.3
10
uM
XMD8-85 HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-17.3
10
uM
XMD8-85 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-12.4
10
uM
XMD8-85 HeLa BARK1
DLkPANILLDEHGHVR
Lys2
-22.1
10
uM
XMD8-85 HeLa BTK
GQYDVAIkMIK
Lys1
-18.0
10
uM
XMD8-85 HeLa CAMK1D
LFAVkCIPK
Lys1
0.7
10
uM
XMD8-85 PC-3 CDK5
DLkPQNLLINR
Lys2
-21.8
10
uM
XMD8-85 HeLa CHK1
DIkPENLLLDER
Lys2
-7.7
10
uM
XMD8-85 HeLa CHK2
DLkPENVLLSSQEEDCLIK
Lys2
16.4
10
uM
XMD8-85 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
30.3
10
uM
XMD8-85 HeLa DGKA
IDPVPNTHPLLVFVNPkSGGK
ATP
-1.9
10
uM
XMD8-85 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
-2.0
10
uM
XMD8-85 HeLa FES
LRADNTLVAVkSCR
Lys1
-9.8
10
uM