XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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  • 1 to 25 of 239 records
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
-63.6
10
uM
XMD8-85 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
81.4
10
uM
XMD8-85 PC-3 AGK
ATVFLNPAACkGK
ATP
4.6
10
uM
XMD8-85 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
-11.0
10
uM
XMD8-85 PC-3 AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
14.3
10
uM
XMD8-85 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
-1.2
10
uM
XMD8-85 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
7.8
10
uM
XMD8-85 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
-23.1
10
uM
XMD8-85 HeLa ATR
FYIMMCkPK
ATP
-18.0
10
uM
XMD8-85 PC-3 ATR
FYIMMCkPK
ATP
5.4
10
uM
XMD8-85 HeLa BRAF
DLkSNNIFLHEDLTVK
Lys2
-9.0
10
uM
XMD8-85 HeLa CaMK1a
LVAIkCIAK
Lys1
-11.7
10
uM
XMD8-85 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
55.2
10
uM
XMD8-85 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
50.6
10
uM
XMD8-85 PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
7.6
10
uM
XMD8-85 PC-3 CDK10
DLkVSNLLMTDK
Lys2
-12.2
10
uM
XMD8-85 PC-3 CDK11,CDK8
DLkPANILVMGEGPER
Lys2
6.2
10
uM
XMD8-85 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
-15.8
10
uM
XMD8-85 PC-3 CDK2
DLkPQNLLINTEGAIK
Lys2
3.3
10
uM
XMD8-85 PC-3 CDK5
NRETHEIVALkR
Lys1
-9.5
10
uM
XMD8-85 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
-2.7
10
uM
XMD8-85 PC-3 CDK9
DMkAANVLITR
Lys2
2.1
10
uM
XMD8-85 PC-3 CHK2
VAIkIISK
Lys1
14.0
10
uM
XMD8-85 PC-3 KC1A
DIkPDNFLMGIGR
Lys2
6.1
10
uM
XMD8-85 PC-3 CK1d,CK1e
DVkPDNFLMGLGKK
Lys2
-12.2
10
uM
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  • 1 to 25 of 239 records