XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
-1.3
 10
uM
XMD8-85 HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
74.4
 10
uM
XMD8-85 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
-8.7
 10
uM
XMD8-85 HeLa PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
1.1
 10
uM
XMD8-85 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
16.2
 10
uM
XMD8-85 PC-3 PITSLRE
DLkTSNLLLSHAGILK
Lys2
17.4
 10
uM
XMD8-85 PC-3 PKCa,PKCb
DLkLDNVMLDSEGHIK
Lys2
-27.9
 10
uM
XMD8-85 HeLa PKD1,PKD2
NIVHCDLkPENVLLASADPFPQVK
Lys2
15.6
 10
uM
XMD8-85 HeLa PKR
DLkPSNIFLVDTK
Lys2
-19.2
 10
uM
XMD8-85 PC-3 PKR
DLkPSNIFLVDTK
Lys2
1.7
 10
uM
XMD8-85 HeLa PRPK
FLSGLELVkQGAEAR
ATP Loop
-2.9
 10
uM
XMD8-85 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
17.9
 10
uM
XMD8-85 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-4.7
 10
uM
XMD8-85 HeLa RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
Lys2
-9.0
 10
uM
XMD8-85 HeLa RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
-27.9
 10
uM
XMD8-85 PC-3 RSK2_domain2
DLkPSNILYVDESGNPESIR
Lys2
64.4
 10
uM
XMD8-85 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
27.9
 10
uM
XMD8-85 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
70.1
 10
uM
XMD8-85 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
-131.3
 10
uM
XMD8-85 HeLa SGK3
FYAVkVLQK
Lys1
-13.9
 10
uM
XMD8-85 HeLa SLK
DLkAGNILFTLDGDIK
Lys2
-13.0
 10
uM
XMD8-85 PC-3 SLK
DLkAGNILFTLDGDIK
Lys2
-5.2
 10
uM
XMD8-85 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
7.0
 10
uM
XMD8-85 PC-3 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
Lys1
3.0
 10
uM
XMD8-85 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
-21.5
 10
uM