XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 HeLa HPK1
DKVSGDLVALkMVK
Lys1
-10.1
10
uM
XMD8-85 HeLa IKKE
SGELVAVkVFNTTSYLRPR
Lys1
-34.8
10
uM
XMD8-85 HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
-0.8
10
uM
XMD8-85 HeLa LATS2
VDTHALYAMkTLR
Lys1
-13.5
10
uM
XMD8-85 HeLa LYN
VAVkTLKPGTMSVQAFLEEANLMK
Lys1
-34.8
10
uM
XMD8-85 PC-3 M3K2
VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
-45.7
10
uM
XMD8-85 HeLa MAP3K5
DIkGDNVLINTYSGVLK
Lys2
-12.2
10
uM
XMD8-85 HeLa MAPKAPK3
KYAVTDDYQLSkQVLGLGVNGK
ATP Loop
-15.8
10
uM
XMD8-85 PC-3 MARK2
EVAVkIIDKTQLNSSSLQK
Lys1
-3.9
10
uM
XMD8-85 PC-3 MARK3,MARK4
EVAIkIIDK
Lys1
-5.9
10
uM
XMD8-85 HeLa MASTL
LYAVkVVK
Lys1
-12.0
10
uM
XMD8-85 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
15.3
10
uM
XMD8-85 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
16.7
10
uM
XMD8-85 HeLa p38a
DLkPSNLAVNEDCELK
Lys2
-25.7
10
uM
XMD8-85 PC-3 p38a
DLkPSNLAVNEDCELK
Lys2
-25.7
10
uM
XMD8-85 HeLa MK14
QELNkTIWEVPER
Other
-19.8
10
uM
XMD8-85 PC-3 MK14
QELNkTIWEVPER
Other
-2.9
10
uM
XMD8-85 HeLa PAN3
VMDPTkILITGK
-7.7
10
uM
XMD8-85 HeLa PEK
DLkPSNIFFTMDDVVK
Lys2
-32.9
10
uM
XMD8-85 PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
9.3
10
uM
XMD8-85 HeLa PIK3CG
KkPLWLEFK
ATP
-13.4
10
uM
XMD8-85 HeLa PKN1
GHFGkVLLSEFRPSGELFAIK
Lys1
-20.5
10
uM
XMD8-85 HeLa PLK1
DLkLGNLFLNEDLEVK
Lys2
2.6
10
uM
XMD8-85 PC-3 ROCK1
kLQLELNQER
Other
-11.7
10
uM
XMD8-85 PC-3 RON
IQCAIkSLSR
Lys1
-0.5
10
uM