JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JWE-035 | PC-3 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 5.6 | 10 | uM |
| JWE-035 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | 17.5 | 10 | uM |
| JWE-035 | PC-3 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | 25.8 | 10 | uM |
| JWE-035 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | 13.3 | 10 | uM |
| JWE-035 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -19.6 | 10 | uM |
| JWE-035 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -2.8 | 10 | uM |
| JWE-035 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | 6.5 | 10 | uM |
| JWE-035 | PC-3 | NEK8 | DLkTQNILLDK | Lys2 | 10.6 | 10 | uM |
| JWE-035 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | -6.0 | 10 | uM |
| JWE-035 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | 15.9 | 10 | uM |
| JWE-035 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -19.5 | 10 | uM |
| JWE-035 | PC-3 | NEK9 | LGDYGLAkK | Activation Loop | 30.0 | 10 | uM |
| JWE-035 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -8.8 | 10 | uM |
| JWE-035 | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -5.8 | 10 | uM |
| JWE-035 | HeLa | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 9.6 | 10 | uM |
| JWE-035 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 2.1 | 10 | uM |
| JWE-035 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | 5.3 | 10 | uM |
| JWE-035 | HeLa | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | 10.9 | 10 | uM |
| JWE-035 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | 2.7 | 10 | uM |
| JWE-035 | HeLa | PCTAIRE2 | DLkPQNLLINEK | Lys2 | -6.6 | 10 | uM |
| JWE-035 | PC-3 | CDK14 | LVALkVIR | Lys1 | 14.6 | 10 | uM |
| JWE-035 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | 2.4 | 10 | uM |
| JWE-035 | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 30.8 | 10 | uM |
| JWE-035 | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 6.8 | 10 | uM |
| JWE-035 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -25.0 | 10 | uM |