XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-50 | HeLa | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | 0.3 | 10 | uM |
XMD11-50 | PC-3 | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | 13.7 | 10 | uM |
XMD11-50 | PC-3 | TAOK2 | DVkAGNILLSEPGLVK | Lys2 | 11.1 | 10 | uM |
XMD11-50 | HeLa | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | 21.4 | 10 | uM |
XMD11-50 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -0.8 | 10 | uM |
XMD11-50 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | 8.2 | 10 | uM |
XMD11-50 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | -0.3 | 10 | uM |
XMD11-50 | HeLa | WEE1 | YIHSMSLVHMDIkPSNIFISR | Lys2 | -17.5 | 10 | uM |
XMD11-50 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | 7.6 | 10 | uM |
XMD11-50 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | 8.4 | 10 | uM |
XMD11-50 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | 1.4 | 10 | uM |
XMD11-50 | HeLa | MLTK | WISQDKEVAVKk | Lys1 | 8.5 | 10 | uM |
XMD11-50 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 3.0 | 10 | uM |
XMD11-50 | HeLa | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -10.9 | 10 | uM |
XMD11-50 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 5.8 | 10 | uM |
XMD11-50 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | 19.6 | 10 | uM |
XMD11-50 | HeLa | BTK | GQYDVAIkMIK | Lys1 | -7.8 | 10 | uM |
XMD11-50 | HeLa | CAMK1D | LFAVkCIPK | Lys1 | 5.4 | 10 | uM |
XMD11-50 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 8.5 | 10 | uM |
XMD11-50 | HeLa | CHK1 | DIkPENLLLDER | Lys2 | -6.4 | 10 | uM |
XMD11-50 | HeLa | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 14.8 | 10 | uM |
XMD11-50 | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 5.0 | 10 | uM |
XMD11-50 | HeLa | DGKA | IDPVPNTHPLLVFVNPkSGGK | ATP | 11.9 | 10 | uM |
XMD11-50 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | -3.9 | 10 | uM |
XMD11-50 | HeLa | FES | LRADNTLVAVkSCR | Lys1 | 7.5 | 10 | uM |