XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
0.3
10
uM
XMD11-50 PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
13.7
10
uM
XMD11-50 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
11.1
10
uM
XMD11-50 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
21.4
10
uM
XMD11-50 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-0.8
10
uM
XMD11-50 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
8.2
10
uM
XMD11-50 PC-3 TLK2
YVAVkIHQLNK
Lys1
-0.3
10
uM
XMD11-50 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-17.5
10
uM
XMD11-50 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
7.6
10
uM
XMD11-50 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
8.4
10
uM
XMD11-50 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
1.4
10
uM
XMD11-50 HeLa MLTK
WISQDKEVAVKk
Lys1
8.5
10
uM
XMD11-50 PC-3 MLTK
WISQDKEVAVKk
Lys1
3.0
10
uM
XMD11-50 HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-10.9
10
uM
XMD11-50 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
5.8
10
uM
XMD11-50 HeLa BARK1
DLkPANILLDEHGHVR
Lys2
19.6
10
uM
XMD11-50 HeLa BTK
GQYDVAIkMIK
Lys1
-7.8
10
uM
XMD11-50 HeLa CAMK1D
LFAVkCIPK
Lys1
5.4
10
uM
XMD11-50 PC-3 CDK5
DLkPQNLLINR
Lys2
8.5
10
uM
XMD11-50 HeLa CHK1
DIkPENLLLDER
Lys2
-6.4
10
uM
XMD11-50 HeLa CHK2
DLkPENVLLSSQEEDCLIK
Lys2
14.8
10
uM
XMD11-50 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
5.0
10
uM
XMD11-50 HeLa DGKA
IDPVPNTHPLLVFVNPkSGGK
ATP
11.9
10
uM
XMD11-50 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
-3.9
10
uM
XMD11-50 HeLa FES
LRADNTLVAVkSCR
Lys1
7.5
10
uM