XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 HeLa HPK1
DKVSGDLVALkMVK
Lys1
0.6
10
uM
XMD11-50 HeLa IKKE
SGELVAVkVFNTTSYLRPR
Lys1
10.9
10
uM
XMD11-50 HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
13.9
10
uM
XMD11-50 HeLa LATS2
VDTHALYAMkTLR
Lys1
8.4
10
uM
XMD11-50 HeLa LYN
VAVkTLKPGTMSVQAFLEEANLMK
Lys1
13.6
10
uM
XMD11-50 PC-3 M3K2
VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
-48.3
10
uM
XMD11-50 HeLa MAP3K5
DIkGDNVLINTYSGVLK
Lys2
3.7
10
uM
XMD11-50 HeLa MAPKAPK3
KYAVTDDYQLSkQVLGLGVNGK
ATP Loop
25.2
10
uM
XMD11-50 PC-3 MARK2
EVAVkIIDKTQLNSSSLQK
Lys1
-13.9
10
uM
XMD11-50 PC-3 MARK3,MARK4
EVAIkIIDK
Lys1
-0.8
10
uM
XMD11-50 HeLa MASTL
LYAVkVVK
Lys1
14.0
10
uM
XMD11-50 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
-5.7
10
uM
XMD11-50 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
-0.5
10
uM
XMD11-50 HeLa p38a
DLkPSNLAVNEDCELK
Lys2
9.7
10
uM
XMD11-50 PC-3 p38a
DLkPSNLAVNEDCELK
Lys2
-4.7
10
uM
XMD11-50 HeLa MK14
QELNkTIWEVPER
Other
-3.7
10
uM
XMD11-50 PC-3 MK14
QELNkTIWEVPER
Other
11.4
10
uM
XMD11-50 HeLa PAN3
VMDPTkILITGK
1.6
10
uM
XMD11-50 HeLa PEK
DLkPSNIFFTMDDVVK
Lys2
-18.8
10
uM
XMD11-50 PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
-8.5
10
uM
XMD11-50 HeLa PIK3CG
KkPLWLEFK
ATP
-10.0
10
uM
XMD11-50 HeLa PKN1
GHFGkVLLSEFRPSGELFAIK
Lys1
22.8
10
uM
XMD11-50 HeLa PLK1
DLkLGNLFLNEDLEVK
Lys2
42.0
10
uM
XMD11-50 PC-3 ROCK1
kLQLELNQER
Other
-4.3
10
uM
XMD11-50 PC-3 RON
IQCAIkSLSR
Lys1
11.4
10
uM