XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-50 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | -11.4 | 10 | uM |
XMD11-50 | HeLa | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | 14.3 | 10 | uM |
XMD11-50 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | 53.0 | 10 | uM |
XMD11-50 | HeLa | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 25.2 | 10 | uM |
XMD11-50 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 41.8 | 10 | uM |
XMD11-50 | PC-3 | PITSLRE | DLkTSNLLLSHAGILK | Lys2 | 3.0 | 10 | uM |
XMD11-50 | PC-3 | PKCa,PKCb | DLkLDNVMLDSEGHIK | Lys2 | -5.6 | 10 | uM |
XMD11-50 | HeLa | PKD1,PKD2 | NIVHCDLkPENVLLASADPFPQVK | Lys2 | 19.1 | 10 | uM |
XMD11-50 | HeLa | PKR | DLkPSNIFLVDTK | Lys2 | -9.2 | 10 | uM |
XMD11-50 | PC-3 | PKR | DLkPSNIFLVDTK | Lys2 | 2.1 | 10 | uM |
XMD11-50 | HeLa | PRPK | FLSGLELVkQGAEAR | ATP Loop | 6.5 | 10 | uM |
XMD11-50 | PC-3 | PRPK | FLSGLELVkQGAEAR | ATP Loop | 8.3 | 10 | uM |
XMD11-50 | PC-3 | ROCK1,ROCK2 | DVkPDNMLLDK | Lys2 | -10.3 | 10 | uM |
XMD11-50 | HeLa | RSK1,RSK2_domain1 | DLkPENILLDEEGHIKLTDFGLSK | Lys2 | 16.5 | 10 | uM |
XMD11-50 | HeLa | RSK2_domain1 | LTDFGLSkESIDHEKK | Activation Loop | -5.3 | 10 | uM |
XMD11-50 | PC-3 | RSK2_domain2 | DLkPSNILYVDESGNPESIR | Lys2 | 68.2 | 10 | uM |
XMD11-50 | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 34.5 | 10 | uM |
XMD11-50 | PC-3 | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 70.0 | 10 | uM |
XMD11-50 | HeLa | RSKL1_domain1 | VLGVIDkVLLVMDTR | Protein Kinase Domain | 35.7 | 10 | uM |
XMD11-50 | HeLa | SGK3 | FYAVkVLQK | Lys1 | -6.0 | 10 | uM |
XMD11-50 | HeLa | SLK | DLkAGNILFTLDGDIK | Lys2 | 4.9 | 10 | uM |
XMD11-50 | PC-3 | SLK | DLkAGNILFTLDGDIK | Lys2 | 21.0 | 10 | uM |
XMD11-50 | HeLa | SMG1 | DTVTIHSVGGTITILPTkTKPK | ATP | 14.1 | 10 | uM |
XMD11-50 | PC-3 | SRC | VAIkTLKPGTMSPEAFLQEAQVMK | Lys1 | 1.6 | 10 | uM |
XMD11-50 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | -10.3 | 10 | uM |