XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
-11.4
10
uM
XMD11-50 HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
14.3
10
uM
XMD11-50 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
53.0
10
uM
XMD11-50 HeLa PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
25.2
10
uM
XMD11-50 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
41.8
10
uM
XMD11-50 PC-3 PITSLRE
DLkTSNLLLSHAGILK
Lys2
3.0
10
uM
XMD11-50 PC-3 PKCa,PKCb
DLkLDNVMLDSEGHIK
Lys2
-5.6
10
uM
XMD11-50 HeLa PKD1,PKD2
NIVHCDLkPENVLLASADPFPQVK
Lys2
19.1
10
uM
XMD11-50 HeLa PKR
DLkPSNIFLVDTK
Lys2
-9.2
10
uM
XMD11-50 PC-3 PKR
DLkPSNIFLVDTK
Lys2
2.1
10
uM
XMD11-50 HeLa PRPK
FLSGLELVkQGAEAR
ATP Loop
6.5
10
uM
XMD11-50 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
8.3
10
uM
XMD11-50 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-10.3
10
uM
XMD11-50 HeLa RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
Lys2
16.5
10
uM
XMD11-50 HeLa RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
-5.3
10
uM
XMD11-50 PC-3 RSK2_domain2
DLkPSNILYVDESGNPESIR
Lys2
68.2
10
uM
XMD11-50 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
34.5
10
uM
XMD11-50 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
70.0
10
uM
XMD11-50 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
35.7
10
uM
XMD11-50 HeLa SGK3
FYAVkVLQK
Lys1
-6.0
10
uM
XMD11-50 HeLa SLK
DLkAGNILFTLDGDIK
Lys2
4.9
10
uM
XMD11-50 PC-3 SLK
DLkAGNILFTLDGDIK
Lys2
21.0
10
uM
XMD11-50 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
14.1
10
uM
XMD11-50 PC-3 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
Lys1
1.6
10
uM
XMD11-50 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
-10.3
10
uM