XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-50 | HeLa | MAP2K3 | DVkPSNVLINK | Lys2 | 0.0 | 10 | uM |
XMD11-50 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -0.2 | 10 | uM |
XMD11-50 | HeLa | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | 0.2 | 10 | uM |
XMD11-50 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | -0.3 | 10 | uM |
XMD11-50 | HeLa | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | 0.3 | 10 | uM |
XMD11-50 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | 0.3 | 10 | uM |
XMD11-50 | HeLa | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -0.4 | 10 | uM |
XMD11-50 | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 0.4 | 10 | uM |
XMD11-50 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | -0.5 | 10 | uM |
XMD11-50 | PC-3 | M3K2,MAP3K3 | DIkGANILR | Lys2 | -0.5 | 10 | uM |
XMD11-50 | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | -0.5 | 10 | uM |
XMD11-50 | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | 0.6 | 10 | uM |
XMD11-50 | PC-3 | SNRK | DLkPENVVFFEK | Lys2 | -0.7 | 10 | uM |
XMD11-50 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | 0.7 | 10 | uM |
XMD11-50 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -0.8 | 10 | uM |
XMD11-50 | PC-3 | MARK3,MARK4 | EVAIkIIDK | Lys1 | -0.8 | 10 | uM |
XMD11-50 | HeLa | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -0.9 | 10 | uM |
XMD11-50 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 0.9 | 10 | uM |
XMD11-50 | HeLa | PIK3CG | KkPLWLEFK | ATP | -10.0 | 10 | uM |
XMD11-50 | HeLa | M3K2,MAP3K3 | DIkGANILR | Lys2 | 10.0 | 10 | uM |
XMD11-50 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 10.1 | 10 | uM |
XMD11-50 | HeLa | MAP3K5,MAP3K6,MAP3K7 | IAIkEIPERDSR | Lys1 | 10.2 | 10 | uM |
XMD11-50 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | -10.3 | 10 | uM |
XMD11-50 | PC-3 | ROCK1,ROCK2 | DVkPDNMLLDK | Lys2 | -10.3 | 10 | uM |
XMD11-50 | PC-3 | ATR | FYIMMCkPK | ATP | -10.3 | 10 | uM |