XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 HeLa MAP2K3
DVkPSNVLINK
Lys2
0.0
10
uM
XMD11-50 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-0.2
10
uM
XMD11-50 HeLa KS6B1
DLkPENIMLNHQGHVK
Lys2
0.2
10
uM
XMD11-50 PC-3 TLK2
YVAVkIHQLNK
Lys1
-0.3
10
uM
XMD11-50 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
0.3
10
uM
XMD11-50 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
0.3
10
uM
XMD11-50 HeLa NEK6,NEK7
DIkPANVFITATGVVK
Lys2
-0.4
10
uM
XMD11-50 PC-3 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
0.4
10
uM
XMD11-50 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
-0.5
10
uM
XMD11-50 PC-3 M3K2,MAP3K3
DIkGANILR
Lys2
-0.5
10
uM
XMD11-50 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
-0.5
10
uM
XMD11-50 HeLa HPK1
DKVSGDLVALkMVK
Lys1
0.6
10
uM
XMD11-50 PC-3 SNRK
DLkPENVVFFEK
Lys2
-0.7
10
uM
XMD11-50 HeLa NEK9
DIkTLNIFLTK
Lys2
0.7
10
uM
XMD11-50 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-0.8
10
uM
XMD11-50 PC-3 MARK3,MARK4
EVAIkIIDK
Lys1
-0.8
10
uM
XMD11-50 HeLa p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-0.9
10
uM
XMD11-50 HeLa BRAF
DLkSNNIFLHEDLTVK
Lys2
0.9
10
uM
XMD11-50 HeLa PIK3CG
KkPLWLEFK
ATP
-10.0
10
uM
XMD11-50 HeLa M3K2,MAP3K3
DIkGANILR
Lys2
10.0
10
uM
XMD11-50 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
10.1
10
uM
XMD11-50 HeLa MAP3K5,MAP3K6,MAP3K7
IAIkEIPERDSR
Lys1
10.2
10
uM
XMD11-50 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
-10.3
10
uM
XMD11-50 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-10.3
10
uM
XMD11-50 PC-3 ATR
FYIMMCkPK
ATP
-10.3
10
uM
  • Page 1 of 10
  • 1 to 25 of 239 records