XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
9.8
10
uM
XMD11-50 HeLa LOK
DLkAGNVLMTLEGDIR
Lys2
9.7
10
uM
XMD11-50 HeLa p38a
DLkPSNLAVNEDCELK
Lys2
9.7
10
uM
XMD11-50 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
96.8
10
uM
XMD11-50 HeLa MAP2K6
DVkPSNVLINALGQVK
Lys2
9.5
10
uM
XMD11-50 PC-3 KC1A
DIkPDNFLMGIGR
Lys2
-9.4
10
uM
XMD11-50 HeLa MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
-9.3
10
uM
XMD11-50 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-9.2
10
uM
XMD11-50 HeLa PKR
DLkPSNIFLVDTK
Lys2
-9.2
10
uM
XMD11-50 HeLa MSK1_domain1
DIkLENILLDSNGHVVLTDFGLSK
Lys2
-90.3
10
uM
XMD11-50 PC-3 MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
8.5
10
uM
XMD11-50 PC-3 CDK5
DLkPQNLLINR
Lys2
8.5
10
uM
XMD11-50 HeLa MLTK
WISQDKEVAVKk
Lys1
8.5
10
uM
XMD11-50 HeLa MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
-8.5
10
uM
XMD11-50 PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
-8.5
10
uM
XMD11-50 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
8.4
10
uM
XMD11-50 HeLa LATS2
VDTHALYAMkTLR
Lys1
8.4
10
uM
XMD11-50 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
8.3
10
uM
XMD11-50 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
8.3
10
uM
XMD11-50 HeLa TLK1
YAAVkIHQLNK
Lys1
8.2
10
uM
XMD11-50 PC-3 M4K3
NVNTGELAAIkVIK
Lys1
8.2
10
uM
XMD11-50 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
8.2
10
uM
XMD11-50 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
8.1
10
uM
XMD11-50 HeLa MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
8.1
10
uM
XMD11-50 HeLa GCN2
LDGCCYAVkR
Lys1
8.0
10
uM
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