XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-50 | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | 11.9 | 10 | uM |
XMD11-50 | HeLa | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 28.4 | 10 | uM |
XMD11-50 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 6.4 | 10 | uM |
XMD11-50 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | 35.0 | 10 | uM |
XMD11-50 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -7.5 | 10 | uM |
XMD11-50 | HeLa | ILK | WQGNDIVVkVLK | Lys1 | 3.0 | 10 | uM |
XMD11-50 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -2.4 | 10 | uM |
XMD11-50 | HeLa | DMPK | DIkPDNILLDR | Lys2 | -11.2 | 10 | uM |
XMD11-50 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -18.4 | 10 | uM |
XMD11-50 | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | 96.8 | 10 | uM |
XMD11-50 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | 1.3 | 10 | uM |
XMD11-50 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 55.3 | 10 | uM |
XMD11-50 | HeLa | ABL,ARG | LMTGDTYTAHAGAkFPIK | Activation Loop | -2.8 | 10 | uM |
XMD11-50 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -0.2 | 10 | uM |
XMD11-50 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | 0.3 | 10 | uM |
XMD11-50 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 10.7 | 10 | uM |
XMD11-50 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 2.8 | 10 | uM |
XMD11-50 | HeLa | ATR | FYIMMCkPK | ATP | 2.5 | 10 | uM |
XMD11-50 | HeLa | ACK | TVSVAVkCLKPDVLSQPEAMDDFIR | Lys1 | 69.0 | 10 | uM |
XMD11-50 | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | 8.1 | 10 | uM |
XMD11-50 | HeLa | BRAF | DLkSNNIFLHEDLTVK | Lys2 | 0.9 | 10 | uM |
XMD11-50 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -1.1 | 10 | uM |
XMD11-50 | HeLa | CaMK1a | LVAIkCIAK | Lys1 | 20.5 | 10 | uM |
XMD11-50 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | 5.0 | 10 | uM |
XMD11-50 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | 15.5 | 10 | uM |