XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 HeLa GCK
DTVTSELAAVkIVK
Lys1
11.9
10
uM
XMD11-50 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
28.4
10
uM
XMD11-50 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
6.4
10
uM
XMD11-50 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
35.0
10
uM
XMD11-50 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-7.5
10
uM
XMD11-50 HeLa ILK
WQGNDIVVkVLK
Lys1
3.0
10
uM
XMD11-50 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-2.4
10
uM
XMD11-50 HeLa DMPK
DIkPDNILLDR
Lys2
-11.2
10
uM
XMD11-50 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-18.4
10
uM
XMD11-50 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
96.8
10
uM
XMD11-50 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
1.3
10
uM
XMD11-50 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
55.3
10
uM
XMD11-50 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
-2.8
10
uM
XMD11-50 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-0.2
10
uM
XMD11-50 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
0.3
10
uM
XMD11-50 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
10.7
10
uM
XMD11-50 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
2.8
10
uM
XMD11-50 HeLa ATR
FYIMMCkPK
ATP
2.5
10
uM
XMD11-50 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
69.0
10
uM
XMD11-50 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
8.1
10
uM
XMD11-50 HeLa BRAF
DLkSNNIFLHEDLTVK
Lys2
0.9
10
uM
XMD11-50 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-1.1
10
uM
XMD11-50 HeLa CaMK1a
LVAIkCIAK
Lys1
20.5
10
uM
XMD11-50 HeLa IRE1
DLkPHNILISMPNAHGK
Lys2
5.0
10
uM
XMD11-50 HeLa IRAK4
DIkSANILLDEAFTAK
Lys2
15.5
10
uM
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  • 1 to 25 of 239 records