XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-50 | HeLa | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | -10.9 | 10 | uM |
XMD11-50 | PC-3 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIkGQNVLLTENAEVK | Lys2 | 5.8 | 10 | uM |
XMD11-50 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | 1.4 | 10 | uM |
XMD11-50 | PC-3 | Wnk1,Wnk2,Wnk4 | IGDLGLATLkR | Activation Loop | 8.4 | 10 | uM |
XMD11-50 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | 7.6 | 10 | uM |
XMD11-50 | HeLa | WEE1 | YIHSMSLVHMDIkPSNIFISR | Lys2 | -17.5 | 10 | uM |
XMD11-50 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | 14.3 | 10 | uM |
XMD11-50 | HeLa | ULK1 | DLkPQNILLSNPAGR | Lys2 | -2.0 | 10 | uM |
XMD11-50 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | -0.3 | 10 | uM |
XMD11-50 | PC-3 | TLK1 | YAAVkIHQLNK | Lys1 | 3.0 | 10 | uM |
XMD11-50 | PC-3 | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | 8.2 | 10 | uM |
XMD11-50 | HeLa | TLK1 | YAAVkIHQLNK | Lys1 | 8.2 | 10 | uM |
XMD11-50 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -0.8 | 10 | uM |
XMD11-50 | HeLa | TEC | YVLDDQYTSSSGAkFPVK | Activation Loop | -9.2 | 10 | uM |
XMD11-50 | HeLa | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | 21.4 | 10 | uM |
XMD11-50 | PC-3 | TAOK2 | DVkAGNILLSEPGLVK | Lys2 | 11.1 | 10 | uM |
XMD11-50 | HeLa | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | 0.3 | 10 | uM |
XMD11-50 | PC-3 | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | 13.7 | 10 | uM |
XMD11-50 | HeLa | SYK | ISDFGLSkALR | Activation Loop | -1.7 | 10 | uM |
XMD11-50 | HeLa | STLK5 | YSVkVLPWLSPEVLQQNLQGYDAK | Activation Loop | -10.3 | 10 | uM |
XMD11-50 | PC-3 | SRPK1/2 | FVAMkVVK | Lys1 | 1.7 | 10 | uM |
XMD11-50 | PC-3 | SRPK1 | IIHTDIkPENILLSVNEQYIR | Lys2 | 2.6 | 10 | uM |
XMD11-50 | PC-3 | SRC | VAIkTLKPGTMSPEAFLQEAQVMK | Lys1 | 1.6 | 10 | uM |
XMD11-50 | PC-3 | SNRK | DLkPENVVFFEK | Lys2 | -0.7 | 10 | uM |
XMD11-50 | HeLa | SMG1 | DTVTIHSVGGTITILPTkTKPK | ATP | 14.1 | 10 | uM |