XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-10.9
10
uM
XMD11-50 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
5.8
10
uM
XMD11-50 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
1.4
10
uM
XMD11-50 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
8.4
10
uM
XMD11-50 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
7.6
10
uM
XMD11-50 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-17.5
10
uM
XMD11-50 HeLa ULK3
EVVAIkCVAK
Lys1
14.3
10
uM
XMD11-50 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-2.0
10
uM
XMD11-50 PC-3 TLK2
YVAVkIHQLNK
Lys1
-0.3
10
uM
XMD11-50 PC-3 TLK1
YAAVkIHQLNK
Lys1
3.0
10
uM
XMD11-50 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
8.2
10
uM
XMD11-50 HeLa TLK1
YAAVkIHQLNK
Lys1
8.2
10
uM
XMD11-50 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-0.8
10
uM
XMD11-50 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-9.2
10
uM
XMD11-50 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
21.4
10
uM
XMD11-50 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
11.1
10
uM
XMD11-50 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
0.3
10
uM
XMD11-50 PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
13.7
10
uM
XMD11-50 HeLa SYK
ISDFGLSkALR
Activation Loop
-1.7
10
uM
XMD11-50 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
-10.3
10
uM
XMD11-50 PC-3 SRPK1/2
FVAMkVVK
Lys1
1.7
10
uM
XMD11-50 PC-3 SRPK1
IIHTDIkPENILLSVNEQYIR
Lys2
2.6
10
uM
XMD11-50 PC-3 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
Lys1
1.6
10
uM
XMD11-50 PC-3 SNRK
DLkPENVVFFEK
Lys2
-0.7
10
uM
XMD11-50 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
14.1
10
uM
  • Page 1 of 10
  • 1 to 25 of 239 records