XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 HeLa RIPK3
DLkPSNVLLDPELHVK
Lys2
5.1
10
uM
XMD11-50 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-20.7
10
uM
XMD11-50 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
17.3
10
uM
XMD11-50 PC-3 SLK
ETSVLAAAkVIDTK
Lys1
1.5
10
uM
XMD11-50 HeLa SYK
ISDFGLSkALR
Activation Loop
-1.7
10
uM
XMD11-50 HeLa TLK1
YAAVkIHQLNK
Lys1
8.2
10
uM
XMD11-50 PC-3 TLK1
YAAVkIHQLNK
Lys1
3.0
10
uM
XMD11-50 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-2.0
10
uM
XMD11-50 HeLa AurB
SHFIVALkVLFK
Lys1
67.9
10
uM
XMD11-50 PC-3 CLK2
LTHTDLkPENILFVNSDYELTYNLEK
Lys2
-22.2
10
uM
XMD11-50 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
7.4
10
uM
XMD11-50 HeLa MYO3A,MYO3B
DVkGNNILLTTEGGVK
Lys2
5.0
10
uM
XMD11-50 PC-3 SNRK
DLkPENVVFFEK
Lys2
-0.7
10
uM
XMD11-50 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-9.2
10
uM