XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-50 PC-3 SRPK1
IIHTDIkPENILLSVNEQYIR
Lys2
2.6
10
uM
XMD11-50 PC-3 SRPK1/2
FVAMkVVK
Lys1
1.7
10
uM
XMD11-50 HeLa ULK3
EVVAIkCVAK
Lys1
14.3
10
uM
XMD11-50 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
1.2
10
uM
XMD11-50 HeLa KPCI
IYAMkVVK
Lys1
20.0
10
uM
XMD11-50 PC-3 PRP4
CNILHADIkPDNILVNESK
Lys2
-11.3
10
uM
XMD11-50 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
-15.2
10
uM
XMD11-50 PC-3 CaMK2a,CaMK2b,CaMK2d,CaMK2g
DLkPENLLLASK
Lys2
61.6
10
uM
XMD11-50 PC-3 CDK5
ETHEIVALkR
Lys1
-3.9
10
uM
XMD11-50 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
2.2
10
uM
XMD11-50 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
-0.5
10
uM
XMD11-50 PC-3 EPHA2
EVPVAIkTLK
Lys1
-15.6
10
uM
XMD11-50 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
13.1
10
uM
XMD11-50 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
-17.2
10
uM
XMD11-50 HeLa GCN2
LDGCCYAVkR
Lys1
8.0
10
uM
XMD11-50 PC-3 GCN2
LDGCCYAVkR
Lys1
1.6
10
uM
XMD11-50 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
9.8
10
uM
XMD11-50 HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
-57.8
10
uM
XMD11-50 PC-3 M4K3
NVNTGELAAIkVIK
Lys1
8.2
10
uM
XMD11-50 PC-3 MET
DMYDKEYYSVHNkTGAK
Activation Loop
-12.5
10
uM
XMD11-50 PC-3 MRCKb
DIkPDNVLLDVNGHIR
Lys2
-16.4
10
uM
XMD11-50 PC-3 MK11
QELNkTVWEVPQR
Other
26.3
10
uM
XMD11-50 PC-3 PDK1
EYAIkILEK
Lys1
11.6
10
uM
XMD11-50 PC-3 PI42C
ELPTLkDMDFLNK
ATP
29.2
10
uM
XMD11-50 HeLa PKD2
DVAVkVIDK
Lys1
6.6
10
uM