XMD11-50 KiNativ -- single dose experiment - Dataset (ID:20097)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-50 | PC-3 | SRPK1 | IIHTDIkPENILLSVNEQYIR | Lys2 | 2.6 | 10 | uM |
XMD11-50 | PC-3 | SRPK1/2 | FVAMkVVK | Lys1 | 1.7 | 10 | uM |
XMD11-50 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | 14.3 | 10 | uM |
XMD11-50 | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | 1.2 | 10 | uM |
XMD11-50 | HeLa | KPCI | IYAMkVVK | Lys1 | 20.0 | 10 | uM |
XMD11-50 | PC-3 | PRP4 | CNILHADIkPDNILVNESK | Lys2 | -11.3 | 10 | uM |
XMD11-50 | PC-3 | ANPb | GMAFLHNSIISSHGSLkSSNCVVDSR | Lys2 | -15.2 | 10 | uM |
XMD11-50 | PC-3 | CaMK2a,CaMK2b,CaMK2d,CaMK2g | DLkPENLLLASK | Lys2 | 61.6 | 10 | uM |
XMD11-50 | PC-3 | CDK5 | ETHEIVALkR | Lys1 | -3.9 | 10 | uM |
XMD11-50 | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | 2.2 | 10 | uM |
XMD11-50 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | -0.5 | 10 | uM |
XMD11-50 | PC-3 | EPHA2 | EVPVAIkTLK | Lys1 | -15.6 | 10 | uM |
XMD11-50 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 13.1 | 10 | uM |
XMD11-50 | PC-3 | EPHB2 | FLEDDTSDPTYTSALGGkIPIR | Activation Loop | -17.2 | 10 | uM |
XMD11-50 | HeLa | GCN2 | LDGCCYAVkR | Lys1 | 8.0 | 10 | uM |
XMD11-50 | PC-3 | GCN2 | LDGCCYAVkR | Lys1 | 1.6 | 10 | uM |
XMD11-50 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | 9.8 | 10 | uM |
XMD11-50 | HeLa | JAK3 domain2 | IADFGLAkLLPLDKDYYVVR | Activation Loop | -57.8 | 10 | uM |
XMD11-50 | PC-3 | M4K3 | NVNTGELAAIkVIK | Lys1 | 8.2 | 10 | uM |
XMD11-50 | PC-3 | MET | DMYDKEYYSVHNkTGAK | Activation Loop | -12.5 | 10 | uM |
XMD11-50 | PC-3 | MRCKb | DIkPDNVLLDVNGHIR | Lys2 | -16.4 | 10 | uM |
XMD11-50 | PC-3 | MK11 | QELNkTVWEVPQR | Other | 26.3 | 10 | uM |
XMD11-50 | PC-3 | PDK1 | EYAIkILEK | Lys1 | 11.6 | 10 | uM |
XMD11-50 | PC-3 | PI42C | ELPTLkDMDFLNK | ATP | 29.2 | 10 | uM |
XMD11-50 | HeLa | PKD2 | DVAVkVIDK | Lys1 | 6.6 | 10 | uM |