Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
A-375 Vemurafenib Methylstat 1.0000 0.5333
uM
48
hr
2 2362 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 141.85 NGFR rabbit IgG(H+L) / donkey NGFR 141.45
A375-B1-rep2
F6
A-375 Vemurafenib I-BET151 1.0000 0.5333
uM
48
hr
2 2401 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 153.82 NGFR rabbit IgG(H+L) / donkey NGFR 109.14
A375-B1-rep2
F7
A-375 Vemurafenib CX-5461 1.0000 0.5333
uM
48
hr
2 1227 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 123.06 NGFR rabbit IgG(H+L) / donkey NGFR 136.57
A375-B1-rep2
F8
A-375 Vemurafenib RG-108 1.0000 0.5333
uM
48
hr
2 1758 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 186.76 NGFR rabbit IgG(H+L) / donkey NGFR 147.11
A375-B1-rep2
G2
A-375 Vemurafenib Anacardic acid 1.0000 0.5333
uM
48
hr
2 1745 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 183.73 NGFR rabbit IgG(H+L) / donkey NGFR 158.90
A375-B1-rep2
G3
A-375 Vemurafenib MC1568 1.0000 0.5333
uM
48
hr
2 2064 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 299.54 NGFR rabbit IgG(H+L) / donkey NGFR 157.98
A375-B1-rep2
G4
A-375 Vemurafenib UNC0638 1.0000 0.5333
uM
48
hr
2 1689 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 178.69 NGFR rabbit IgG(H+L) / donkey NGFR 113.11
A375-B1-rep2
G5
A-375 Vemurafenib Tranylcypromine 1.0000 0.5333
uM
48
hr
2 1765 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 166.51 NGFR rabbit IgG(H+L) / donkey NGFR 168.79
A375-B1-rep2
G6
A-375 Vemurafenib Ischemin 1.0000 0.5333
uM
48
hr
2 1846 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 204.07 NGFR rabbit IgG(H+L) / donkey NGFR 168.74
A375-B1-rep2
G7
A-375 Vemurafenib 1.0000
uM
48
hr
2 1429 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 185.39 NGFR rabbit IgG(H+L) / donkey NGFR 144.00
A375-B1-rep2
H10
A-375 Vemurafenib 1.0000
uM
48
hr
2 1364 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 201.35 NGFR rabbit IgG(H+L) / donkey NGFR 138.83
A375-B1-rep2
H11
A-375 Vemurafenib 1.0000
uM
48
hr
2 1542 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 194.78 NGFR rabbit IgG(H+L) / donkey NGFR 167.11
A375-B1-rep2
H2
A-375 Vemurafenib 1.0000
uM
48
hr
2 1421 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 197.45 NGFR rabbit IgG(H+L) / donkey NGFR 159.25
A375-B1-rep2
H3
A-375 Vemurafenib 1.0000
uM
48
hr
2 1303 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 204.72 NGFR rabbit IgG(H+L) / donkey NGFR 152.30
A375-B1-rep2
H4
A-375 Vemurafenib 1.0000
uM
48
hr
2 1126 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 214.28 NGFR rabbit IgG(H+L) / donkey NGFR 175.81
A375-B1-rep2
H5
A-375 Vemurafenib 1.0000
uM
48
hr
2 1114 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 185.61 NGFR rabbit IgG(H+L) / donkey NGFR 154.43
A375-B1-rep2
H6
A-375 Vemurafenib 1.0000
uM
48
hr
2 1100 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 184.49 NGFR rabbit IgG(H+L) / donkey NGFR 149.00
A375-B1-rep2
H7
A-375 Vemurafenib 1.0000
uM
48
hr
2 1159 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 193.23 NGFR rabbit IgG(H+L) / donkey NGFR 133.62
A375-B1-rep2
H8
A-375 Vemurafenib 1.0000
uM
48
hr
2 1248 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 183.32 NGFR rabbit IgG(H+L) / donkey NGFR 137.61
A375-B1-rep2
H9
A-375 Vemurafenib 1.0000
uM
48
hr
1 2268 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 202.77 NGFR rabbit IgG(H+L) / donkey NGFR 187.51
A375-B2-rep1
A10
A-375 Vemurafenib 1.0000
uM
48
hr
1 2280 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 223.55 NGFR rabbit IgG(H+L) / donkey NGFR 187.85
A375-B2-rep1
A11
A-375 Vemurafenib 1.0000
uM
48
hr
1 2478 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 193.11 NGFR rabbit IgG(H+L) / donkey NGFR 175.65
A375-B2-rep1
A2
A-375 Vemurafenib 1.0000
uM
48
hr
1 2443 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 184.77 NGFR rabbit IgG(H+L) / donkey NGFR 168.94
A375-B2-rep1
A3
A-375 Vemurafenib 1.0000
uM
48
hr
1 2754 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 179.51 NGFR rabbit IgG(H+L) / donkey NGFR 205.98
A375-B2-rep1
A4
A-375 Vemurafenib 1.0000
uM
48
hr
1 2345 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 172.31 NGFR rabbit IgG(H+L) / donkey NGFR 193.43
A375-B2-rep1
A5