Growth rate-corrected (GR) dose-response metrics across a panel of 71 breast cancer cell lines treated with a library of small molecule and antibody perturbagens. Dataset 1 of 4: Relative cell counts and normalized growth rate inhibition values across technical replicates. - Dataset (ID:20268)

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Cell Clinical Subtype Transcriptional Subtype Small Molecule Antibody Perturbagen Target Perturbagen Class Perturbagen Concentration Perturbagen Conc Unit Biological Replicate ID Relative Cell Count Normalized Growth Rate Inhibition Value Nominal Division Rate
184A1
NM
Basal
(Z)-4-Hydroxytamoxifen
ESR1
0.0107
uM
9047.132
0.8736 0.6481 0.6985
184A1
NM
Basal
5-FU
TYMS
TYMS
769
uM
9047.017
0.1559 -0.7788 0.8440
184A1
NM
Basal
5-FU
TYMS
TYMS
19200
uM
9047.017
0.1196 -0.8384 0.8440
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
0.000171
uM
12509.165
0.9871 0.9828 1.5022
184A1
NM
Basal
(Z)-4-Hydroxytamoxifen
ESR1
6.67
uM
9047.132
0.8373 0.5511 0.6985
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
0.533
uM
12509.165
0.3318 -0.0404 1.5022
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
0.107
uM
12509.165
0.3373 -0.0298 1.5022
184A1
NM
Basal
AS-252424
PI3K
PI3K
0.0000853
uM
12509.165
1.0144 1.0191 1.5022
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
13.3
uM
12509.165
0.0484 -0.7335 1.5022
184A1
NM
Basal
AS-252424
PI3K
PI3K
0.0107
uM
12509.165
0.9308 0.9067 1.5022
184A1
NM
Basal
Afatinib
EGFR/HER2
ErbB
2.67
uM
12509.165
0.3136 -0.0757 1.5022
184A1
NM
Basal
AS-252424
PI3K
PI3K
0.267
uM
12509.165
0.8921 0.8536 1.5022
184A1
NM
Basal
(Z)-4-Hydroxytamoxifen
ESR1
33.3
uM
9047.132
0.7816 0.4055 0.6985
184A1
NM
Basal
17-AAG
HSP90
HSP90
100
uM
9047.037
0.0825 -0.9826 0.5262
184A1
NM
Basal
5-DFUR
TYMS
TYMS
1.6
uM
12509.143
1.0174 1.0259 1.3392
184A1
NM
Basal
17-AAG
HSP90
HSP90
0.16
uM
9047.037
0.4280 -0.6013 0.5262
184A1
NM
Basal
(Z)-4-Hydroxytamoxifen
ESR1
0.0533
uM
9047.132
0.9788 0.9394 0.6985
184A1
NM
Basal
17-AAG
HSP90
HSP90
0.000256
uM
9047.037
0.9096 0.6705 0.5262
184A1
NM
Basal
17-AAG
HSP90
HSP90
0.0064
uM
9047.037
0.9396 0.7765 0.5262
184A1
NM
Basal
17-AAG
HSP90
HSP90
0.00128
uM
9047.037
1.0758 1.2981 0.5262
184A1
NM
Basal
(Z)-4-Hydroxytamoxifen
ESR1
167
uM
9047.132
0.9698 0.9141 0.6985
184A1
NM
Basal
17-AAG
HSP90
HSP90
4
uM
9047.037
0.4226 -0.6108 0.5262
184A1
NM
Basal
17-AAG
HSP90
HSP90
0.8
uM
9047.037
0.4311 -0.5959 0.5262
184A1
NM
Basal
Baicalein
Lipoxygenase
Metabolism
0.0107
uM
5895.073
1.0510 1.0702 1.4431
184A1
NM
Basal
Baicalein
Lipoxygenase
Metabolism
0.00213
uM
5895.073
1.0337 1.0465 1.4431