Growth rate-corrected (GR) dose-response metrics across a panel of 71 breast cancer cell lines treated with a library of small molecule and antibody perturbagens. Dataset 1 of 4: Relative cell counts and normalized growth rate inhibition values across technical replicates. - Dataset (ID:20268)
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Cell | Clinical Subtype | Transcriptional Subtype | Small Molecule | Antibody | Perturbagen Target | Perturbagen Class | Perturbagen Concentration | Perturbagen Conc Unit | Biological Replicate ID | Relative Cell Count | Normalized Growth Rate Inhibition Value | Nominal Division Rate |
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184A1 | NM | Basal | (Z)-4-Hydroxytamoxifen | ESR1 | 0.0107 | uM | 9047.132 | 0.8736 | 0.6481 | 0.6985 | ||
184A1 | NM | Basal | 5-FU | TYMS | TYMS | 769 | uM | 9047.017 | 0.1559 | -0.7788 | 0.8440 | |
184A1 | NM | Basal | 5-FU | TYMS | TYMS | 19200 | uM | 9047.017 | 0.1196 | -0.8384 | 0.8440 | |
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 0.000171 | uM | 12509.165 | 0.9871 | 0.9828 | 1.5022 | |
184A1 | NM | Basal | (Z)-4-Hydroxytamoxifen | ESR1 | 6.67 | uM | 9047.132 | 0.8373 | 0.5511 | 0.6985 | ||
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 0.533 | uM | 12509.165 | 0.3318 | -0.0404 | 1.5022 | |
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 0.107 | uM | 12509.165 | 0.3373 | -0.0298 | 1.5022 | |
184A1 | NM | Basal | AS-252424 | PI3K | PI3K | 0.0000853 | uM | 12509.165 | 1.0144 | 1.0191 | 1.5022 | |
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 13.3 | uM | 12509.165 | 0.0484 | -0.7335 | 1.5022 | |
184A1 | NM | Basal | AS-252424 | PI3K | PI3K | 0.0107 | uM | 12509.165 | 0.9308 | 0.9067 | 1.5022 | |
184A1 | NM | Basal | Afatinib | EGFR/HER2 | ErbB | 2.67 | uM | 12509.165 | 0.3136 | -0.0757 | 1.5022 | |
184A1 | NM | Basal | AS-252424 | PI3K | PI3K | 0.267 | uM | 12509.165 | 0.8921 | 0.8536 | 1.5022 | |
184A1 | NM | Basal | (Z)-4-Hydroxytamoxifen | ESR1 | 33.3 | uM | 9047.132 | 0.7816 | 0.4055 | 0.6985 | ||
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 100 | uM | 9047.037 | 0.0825 | -0.9826 | 0.5262 | |
184A1 | NM | Basal | 5-DFUR | TYMS | TYMS | 1.6 | uM | 12509.143 | 1.0174 | 1.0259 | 1.3392 | |
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 0.16 | uM | 9047.037 | 0.4280 | -0.6013 | 0.5262 | |
184A1 | NM | Basal | (Z)-4-Hydroxytamoxifen | ESR1 | 0.0533 | uM | 9047.132 | 0.9788 | 0.9394 | 0.6985 | ||
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 0.000256 | uM | 9047.037 | 0.9096 | 0.6705 | 0.5262 | |
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 0.0064 | uM | 9047.037 | 0.9396 | 0.7765 | 0.5262 | |
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 0.00128 | uM | 9047.037 | 1.0758 | 1.2981 | 0.5262 | |
184A1 | NM | Basal | (Z)-4-Hydroxytamoxifen | ESR1 | 167 | uM | 9047.132 | 0.9698 | 0.9141 | 0.6985 | ||
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 4 | uM | 9047.037 | 0.4226 | -0.6108 | 0.5262 | |
184A1 | NM | Basal | 17-AAG | HSP90 | HSP90 | 0.8 | uM | 9047.037 | 0.4311 | -0.5959 | 0.5262 | |
184A1 | NM | Basal | Baicalein | Lipoxygenase | Metabolism | 0.0107 | uM | 5895.073 | 1.0510 | 1.0702 | 1.4431 | |
184A1 | NM | Basal | Baicalein | Lipoxygenase | Metabolism | 0.00213 | uM | 5895.073 | 1.0337 | 1.0465 | 1.4431 |