DCC-2036 KiNativ -- single dose experiment - Dataset (ID:20210)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
DCC-2036 | Ramos (RA 1) | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | -15.1 | 1 | uM |
DCC-2036 | Ramos (RA 1) | NEK7 | AACLLDGVPVALKK | Lys1 | 1.6 | 1 | uM |
DCC-2036 | Ramos (RA 1) | KPCI | DLKLDNVLLDSEGHIK | Lys2 | -16.0 | 1 | uM |
DCC-2036 | Ramos (RA 1) | MARK1,MARK2 | EVAVKIIDK | Lys1 | -16.2 | 1 | uM |
DCC-2036 | Ramos (RA 1) | PKD2 | DVAVKVIDK | Lys1 | -16.8 | 1 | uM |
DCC-2036 | Ramos (RA 1) | M3K2,MAP3K3 | DIKGANILR | Lys2 | -16.8 | 1 | uM |
DCC-2036 | Ramos (RA 1) | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | -16.9 | 1 | uM |
DCC-2036 | Ramos (RA 1) | FYV1 | GGKSGAAFYATEDDRFILK | ATP | 16.9 | 1 | uM |
DCC-2036 | Ramos (RA 1) | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | 1.7 | 1 | uM |
DCC-2036 | Ramos (RA 1) | BRAF | DLKSNNIFLHEDLTVK | Lys2 | -17.0 | 1 | uM |
DCC-2036 | Ramos (RA 1) | MK01 | DLKPSNLLLNTTCDLK | Lys2 | -17.9 | 1 | uM |
DCC-2036 | Ramos (RA 1) | STLK6 | SIKASHILISGDGLVTLSGLSHLHSLVK | Lys2 | -1.8 | 1 | uM |
DCC-2036 | Ramos (RA 1) | HPK1 | DKVSGDLVALKMVK | Lys1 | 1.8 | 1 | uM |
DCC-2036 | Ramos (RA 1) | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 18.5 | 1 | uM |
DCC-2036 | Ramos (RA 1) | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | 19.0 | 1 | uM |
DCC-2036 | Ramos (RA 1) | JAK1_domain2 | YDPEGDNTGEQVAVKSLKPESGGNHIADLKK | Lys1 | 19.3 | 1 | uM |
DCC-2036 | Ramos (RA 1) | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | -19.6 | 1 | uM |
DCC-2036 | Ramos (RA 1) | ROCK1,ROCK2 | DVKPDNMLLDK | Lys2 | -19.9 | 1 | uM |
DCC-2036 | Ramos (RA 1) | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 20.1 | 1 | uM |
DCC-2036 | Ramos (RA 1) | KC1A | DIKPDNFLMGIGR | Lys2 | 20.6 | 1 | uM |
DCC-2036 | Ramos (RA 1) | MAP2K6 | DVKPSNVLINALGQVK | Lys2 | -2.1 | 1 | uM |
DCC-2036 | Ramos (RA 1) | MST1 | ETGQIVAIKQVPVESDLQEIIK | Lys1 | -2.1 | 1 | uM |
DCC-2036 | Ramos (RA 1) | ATR | FYIMMCKPK | ATP | 21.3 | 1 | uM |
DCC-2036 | Ramos (RA 1) | FER | TSVAVKTCKEDLPQELK | Lys1 | -21.4 | 1 | uM |
DCC-2036 | Ramos (RA 1) | MK03 | DLKPSNLLINTTCDLK | Lys2 | 2.2 | 1 | uM |