PCI-32765 KiNativ -- single dose experiment - Dataset (ID:20206)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
Ibrutinib | Ramos (RA 1) | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | 54.8 | 1 | uM |
Ibrutinib | Ramos (RA 1) | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | 0.3 | 1 | uM |
Ibrutinib | Ramos (RA 1) | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 7.8 | 1 | uM |
Ibrutinib | Ramos (RA 1) | FYV1 | GGKSGAAFYATEDDRFILK | ATP | -1.5 | 1 | uM |
Ibrutinib | Ramos (RA 1) | GCK | DIKGANLLLTLQGDVK | Lys2 | -5.5 | 1 | uM |
Ibrutinib | Ramos (RA 1) | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 0.1 | 1 | uM |
Ibrutinib | Ramos (RA 1) | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | 8.9 | 1 | uM |
Ibrutinib | Ramos (RA 1) | HPK1 | DKVSGDLVALKMVK | Lys1 | -39.4 | 1 | uM |
Ibrutinib | Ramos (RA 1) | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | 9.6 | 1 | uM |
Ibrutinib | Ramos (RA 1) | IKKE,TBK1 | DIKPGNIMR | Lys2 | -66.6 | 1 | uM |
Ibrutinib | Ramos (RA 1) | ILK | ISMADVKFSFQCPGR | Protein Kinase Domain | -37.6 | 1 | uM |
Ibrutinib | Ramos (RA 1) | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 5.7 | 1 | uM |
Ibrutinib | Ramos (RA 1) | JAK1 | QLASALSYLEDKDLVHGNVCTKNLLLAR | Protein Kinase Domain | -61.4 | 1 | uM |
Ibrutinib | Ramos (RA 1) | JAK1_domain2 | YDPEGDNTGEQVAVKSLKPESGGNHIADLKK | Lys1 | -24.2 | 1 | uM |
Ibrutinib | Ramos (RA 1) | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | -3.3 | 1 | uM |
Ibrutinib | Ramos (RA 1) | KC1A | DIKPDNFLMGIGR | Lys2 | -61.7 | 1 | uM |
Ibrutinib | Ramos (RA 1) | KC1G1 | DVKPENFLIGR | Lys2 | -1.8 | 1 | uM |
Ibrutinib | Ramos (RA 1) | KC1G2 | DVKPENFLVGRPGTK | Lys2 | -17.8 | 1 | uM |
Ibrutinib | Ramos (RA 1) | KCC2D | IPTGQEYAAKIINTKK | Lys1 | 24.6 | 1 | uM |
Ibrutinib | Ramos (RA 1) | KCC4 | DLKPENLLYATPAPDAPLK | Lys2 | -3.0 | 1 | uM |
Ibrutinib | Ramos (RA 1) | KHS1 | NVHTGELAAVKIIK | Lys1 | 14.5 | 1 | uM |
Ibrutinib | Ramos (RA 1) | KPCI | DLKLDNVLLDSEGHIK | Lys2 | 19.2 | 1 | uM |
Ibrutinib | Ramos (RA 1) | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | -47.3 | 1 | uM |
Ibrutinib | Ramos (RA 1) | LCK | EGAKFPIKWTAPEAINYGTFTIK | Activation Loop | -2.6 | 1 | uM |
Ibrutinib | Ramos (RA 1) | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | -6.9 | 1 | uM |