QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 BCWM.1 CAMK1D
LFAVKCIPK
Lys1
0.033712822
1
uM
QL-XII-47 BCWM.1 CaMK2g
TSTQEYAAKIINTK
Lys1
4.50076179
1
uM
QL-XII-47 MWCL.1 CaMK2g
TSTQEYAAKIINTK
Lys1
-11.28758926
1
uM
QL-XII-47 MWCL.1 CaMKK2
DIKPSNLLVGEDGHIK
Lys2
11.9973621
1
uM
QL-XII-47 BCWM.1 CaMKK2
DIKPSNLLVGEDGHIK
Lys2
11.88734459
1
uM
QL-XII-47 MWCL.1 CASK
ETGQQFAVKIVDVAK
Lys1
20.5361767
1
uM
QL-XII-47 BCWM.1 CASK
ETGQQFAVKIVDVAK
Lys1
32.90610469
1
uM
QL-XII-47 BCWM.1 CDC2
DLKPQNLLIDDKGTIK
Lys2
-11.32754424
1
uM
QL-XII-47 MWCL.1 CDC2
DLKPQNLLIDDKGTIK
Lys2
-11.26471968
1
uM
QL-XII-47 MWCL.1 CDK11,CDK8
DLKPANILVMGEGPER
Lys2
4.501665604
1
uM
QL-XII-47 BCWM.1 CDK11,CDK8
DLKPANILVMGEGPER
Lys2
14.74034939
1
uM
QL-XII-47 MWCL.1 CDK14
LVALKVIR
Lys1
11.18847664
1
uM
QL-XII-47 BCWM.1 CDK14
LVALKVIR
Lys1
20.63298661
1
uM
QL-XII-47 MWCL.1 CDK16
SKLTDNLVALKEIR
Lys1
15.03393916
1
uM
QL-XII-47 BCWM.1 CDK16
SKLTDNLVALKEIR
Lys1
29.54620403
1
uM
QL-XII-47 BCWM.1 CDK2
DLKPQNLLINTEGAIK
Lys2
-1.556399301
1
uM
QL-XII-47 MWCL.1 CDK2
DLKPQNLLINTEGAIK
Lys2
-3.151747592
1
uM
QL-XII-47 BCWM.1 CDK4
DLKPENILVTSGGTVK
Lys2
-9.229049081
1
uM
QL-XII-47 MWCL.1 CDK4
DLKPENILVTSGGTVK
Lys2
-6.2228303
1
uM
QL-XII-47 BCWM.1 CDK5
DLKPQNLLINR
Lys2
4.004453656
1
uM
QL-XII-47 MWCL.1 CDK5
DLKPQNLLINR
Lys2
-8.984027957
1
uM
QL-XII-47 BCWM.1 CDK6
DLKPQNILVTSSGQIK
Lys2
-0.544166997
1
uM
QL-XII-47 MWCL.1 CDK6
DLKPQNILVTSSGQIK
Lys2
3.69039298
1
uM
QL-XII-47 BCWM.1 CDK7
DLKPNNLLLDENGVLK
Lys2
15.31231831
1
uM
QL-XII-47 MWCL.1 CDK7
DLKPNNLLLDENGVLK
Lys2
17.57459374
1
uM