QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | BCWM.1 | NEK8 | DLKTQNILLDK | Lys2 | 9.444227339 | 1 | uM |
QL-XII-47 | MWCL.1 | NEK8 | DLKTQNILLDK | Lys2 | -11.66656364 | 1 | uM |
QL-XII-47 | BCWM.1 | NEK9 | DIKTLNIFLTK | Lys2 | -8.692345813 | 1 | uM |
QL-XII-47 | MWCL.1 | NEK9 | DIKTLNIFLTK | Lys2 | 5.459866538 | 1 | uM |
QL-XII-47 | MWCL.1 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | -3.9708776 | 1 | uM |
QL-XII-47 | BCWM.1 | OSR1 | DVKAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | -2.037568348 | 1 | uM |
QL-XII-47 | MWCL.1 | p38a | DLKPSNLAVNEDCELK | Lys2 | -6.02251032 | 1 | uM |
QL-XII-47 | BCWM.1 | p38a | DLKPSNLAVNEDCELK | Lys2 | -8.718461078 | 1 | uM |
QL-XII-47 | BCWM.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | 1.738509549 | 1 | uM |
QL-XII-47 | MWCL.1 | p38d,p38g | DLKPGNLAVNEDCELK | Lys2 | -22.53478157 | 1 | uM |
QL-XII-47 | BCWM.1 | PAN3 | VMDPTKILITGK | ATP | 34.20265652 | 1 | uM |
QL-XII-47 | MWCL.1 | PAN3 | VMDPTKILITGK | ATP | 9.049225166 | 1 | uM |
QL-XII-47 | MWCL.1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | 14.83800488 | 1 | uM |
QL-XII-47 | BCWM.1 | PCTAIRE2,PCTAIRE3 | SKLTENLVALKEIR | Lys1 | -7.31403483 | 1 | uM |
QL-XII-47 | BCWM.1 | PDK1 | EYAIKILEK | Lys1 | -13.88134428 | 1 | uM |
QL-XII-47 | MWCL.1 | PDK1 | EYAIKILEK | Lys1 | 15.62608754 | 1 | uM |
QL-XII-47 | BCWM.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | 11.19892963 | 1 | uM |
QL-XII-47 | MWCL.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | -14.59790065 | 1 | uM |
QL-XII-47 | BCWM.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | 22.98766626 | 1 | uM |
QL-XII-47 | MWCL.1 | PHKg2 | ATGHEFAVKIMEVTAER | Lys1 | ND | 1 | uM |
QL-XII-47 | BCWM.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | 4.443788957 | 1 | uM |
QL-XII-47 | MWCL.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | 2.368941706 | 1 | uM |
QL-XII-47 | BCWM.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | 3.960959449 | 1 | uM |
QL-XII-47 | MWCL.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | -2.074607939 | 1 | uM |
QL-XII-47 | BCWM.1 | PI4KB | VPHTQAVVLNSKDK | ATP | 7.838958764 | 1 | uM |