QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | BCWM.1 | NEK3 | SKNIFLTQNGK | Activation Loop | -10.13654488 | 1 | uM |
QL-XII-47 | MWCL.1 | SLK | DLKAGNILFTLDGDIK | Lys2 | 1.020533171 | 1 | uM |
QL-XII-47 | MWCL.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | -1.027450805 | 1 | uM |
QL-XII-47 | MWCL.1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 10.33171657 | 1 | uM |
QL-XII-47 | BCWM.1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | 10.38740966 | 1 | uM |
QL-XII-47 | BCWM.1 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | 10.43573458 | 1 | uM |
QL-XII-47 | MWCL.1 | KHS1 | NVHTGELAAVKIIK | Lys1 | 10.44210585 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP2K1 | IMHRDVKPSNILVNSR | Lys2 | -10.45585154 | 1 | uM |
QL-XII-47 | MWCL.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 10.48021172 | 1 | uM |
QL-XII-47 | MWCL.1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | -10.55702775 | 1 | uM |
QL-XII-47 | MWCL.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | 10.94267365 | 1 | uM |
QL-XII-47 | BCWM.1 | ILK | WQGNDIVVKVLK | Lys1 | 1.096021819 | 1 | uM |
QL-XII-47 | MWCL.1 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | -11.09760984 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP2K3 | DVKPSNVLINK | Lys2 | -11.1285874 | 1 | uM |
QL-XII-47 | MWCL.1 | CDK14 | LVALKVIR | Lys1 | 11.18847664 | 1 | uM |
QL-XII-47 | BCWM.1 | PEK | DLKPSNIFFTMDDVVK | Lys2 | 11.19892963 | 1 | uM |
QL-XII-47 | MWCL.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -11.26471968 | 1 | uM |
QL-XII-47 | MWCL.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | -11.28758926 | 1 | uM |
QL-XII-47 | BCWM.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -11.32754424 | 1 | uM |
QL-XII-47 | MWCL.1 | AurA | FILALKVLFK | Lys1 | 11.33219394 | 1 | uM |
QL-XII-47 | MWCL.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | -11.39063633 | 1 | uM |
QL-XII-47 | BCWM.1 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 11.52268187 | 1 | uM |
QL-XII-47 | MWCL.1 | FYV1 | GGKSGAAFYATEDDRFILK | ATP | 11.54045713 | 1 | uM |
QL-XII-47 | BCWM.1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | -1.155961788 | 1 | uM |
QL-XII-47 | BCWM.1 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | 1.156231522 | 1 | uM |