QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | BCWM.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 4.50076179 | 1 | uM |
QL-XII-47 | MWCL.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 4.501665604 | 1 | uM |
QL-XII-47 | BCWM.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | 4.534711447 | 1 | uM |
QL-XII-47 | MWCL.1 | PIK3CD | VNWLAHNVSKDNRQ | ATP | 4.546978964 | 1 | uM |
QL-XII-47 | MWCL.1 | MP2K7 | DVKPSNILLDER | Lys2 | -45.5174114 | 1 | uM |
QL-XII-47 | BCWM.1 | LATS1 | ALYATKTLR | Lys1 | 4.639137919 | 1 | uM |
QL-XII-47 | BCWM.1 | RSKL1_domain1 | VLGVIDKVLLVMDTR | ATP | 46.48841594 | 1 | uM |
QL-XII-47 | MWCL.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.6555368 | 1 | uM |
QL-XII-47 | BCWM.1 | MSK2 domain1 | DLKLENVLLDSEGHIVLTDFGLSK | Lys2 | -46.59383779 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP2K4 | DIKPSNILLDR | Lys2 | -4.661208852 | 1 | uM |
QL-XII-47 | BCWM.1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | -4.698942545 | 1 | uM |
QL-XII-47 | BCWM.1 | BLK | IIDSEYTAQEGAKFPIK | Activation Loop | 47.0732956 | 1 | uM |
QL-XII-47 | BCWM.1 | MST4 | TQQVVAIKIIDLEEAEDEIEDIQQEITVLSQCDSSYVTK | Lys1 | 4.712110007 | 1 | uM |
QL-XII-47 | BCWM.1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | -4.774099061 | 1 | uM |
QL-XII-47 | MWCL.1 | RSK2 domain1 | DLKPENILLDEEGHIKLTDFGLSKESIDHEK | Lys2 | -48.46241013 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP3K7,TAK1 | DLKPPNLLLVAGGTVLK | Lys2 | 4.848341421 | 1 | uM |
QL-XII-47 | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.884271122 | 1 | uM |
QL-XII-47 | BCWM.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | -4.886038638 | 1 | uM |
QL-XII-47 | BCWM.1 | ITPK1 | ESIFFNSHNVSKPESSSVLTELDKIEGVFERPSDEVIR | ATP | 49.00978471 | 1 | uM |
QL-XII-47 | MWCL.1 | MASTL | LYAVKVVK | Lys1 | -4.9183009 | 1 | uM |
QL-XII-47 | BCWM.1 | PIK3CG | KKPLWLEFK | ATP | -49.28259781 | 1 | uM |
QL-XII-47 | MWCL.1 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | -49.83844146 | 1 | uM |
QL-XII-47 | BCWM.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | -49.97672913 | 1 | uM |
QL-XII-47 | MWCL.1 | RIPK2 | VQVAVKHLHIHTPLLDSER | Lys1 | 5.017497496 | 1 | uM |
QL-XII-47 | MWCL.1 | KC1A | DIKPDNFLMGIGR | Lys2 | -5.104906235 | 1 | uM |