QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | BCWM.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 2.746888981 | 1 | uM |
| QL-XII-47 | MWCL.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | -1.027450805 | 1 | uM |
| QL-XII-47 | BCWM.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | -24.56149352 | 1 | uM |
| QL-XII-47 | BCWM.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | -59.65168038 | 1 | uM |
| QL-XII-47 | MWCL.1 | NEK3 | SKNIFLTQNGK | Activation Loop | 9.919741065 | 1 | uM |
| QL-XII-47 | MWCL.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | -4.6555368 | 1 | uM |
| QL-XII-47 | MWCL.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | -87.4730226 | 1 | uM |
| QL-XII-47 | MWCL.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | -9.341503001 | 1 | uM |
| QL-XII-47 | BCWM.1 | NEK3 | SKNIFLTQNGK | Activation Loop | -10.13654488 | 1 | uM |
| QL-XII-47 | BCWM.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | -37.08301629 | 1 | uM |
| QL-XII-47 | MWCL.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | -18.8674785 | 1 | uM |
| QL-XII-47 | MWCL.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | -17.85533882 | 1 | uM |
| QL-XII-47 | MWCL.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | -8.174014716 | 1 | uM |
| QL-XII-47 | MWCL.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | -31.93905936 | 1 | uM |
| QL-XII-47 | MWCL.1 | DNAPK | KGGSWIQEINVAEK | ATP | 14.36767264 | 1 | uM |
| QL-XII-47 | MWCL.1 | DNAPK | EHPFLVKGGEDLR | ATP | -17.02227611 | 1 | uM |
| QL-XII-47 | MWCL.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | -20.94285661 | 1 | uM |
| QL-XII-47 | BCWM.1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | -4.698942545 | 1 | uM |
| QL-XII-47 | BCWM.1 | DNAPK | EHPFLVKGGEDLR | ATP | -8.763473644 | 1 | uM |
| QL-XII-47 | BCWM.1 | DNAPK | KGGSWIQEINVAEK | ATP | -13.80369189 | 1 | uM |
| QL-XII-47 | BCWM.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | PAN3 | VMDPTKILITGK | ATP | 9.049225166 | 1 | uM |
| QL-XII-47 | MWCL.1 | ATR | FYIMMCKPK | ATP | 26.45300257 | 1 | uM |
| QL-XII-47 | MWCL.1 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | -2.074607939 | 1 | uM |