QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-XII-47 MWCL.1 LKB1
DIKPGNLLLTTGGTLK
Lys2
5.905585783
1
uM
QL-XII-47 MWCL.1 LOK
DLKAGNVLMTLEGDIR
Lys2
-3.152905014
1
uM
QL-XII-47 MWCL.1 LRRK2
DLKPHNVLLFTLYPNAAIIAK
Lys2
7.098641111
1
uM
QL-XII-47 MWCL.1 LYN
VAVKTLKPGTMSVQAFLEEANLMK
Lys1
2.528406343
1
uM
QL-XII-47 MWCL.1 MAP2K1
IMHRDVKPSNILVNSR
Lys2
-10.45585154
1
uM
QL-XII-47 MWCL.1 MAP2K1,MAP2K2
DVKPSNILVNSR
Lys2
2.14775294
1
uM
QL-XII-47 MWCL.1 MAP2K3
DVKPSNVLINK
Lys2
-11.1285874
1
uM
QL-XII-47 MWCL.1 MAP2K4
DIKPSNILLDR
Lys2
-4.661208852
1
uM
QL-XII-47 MWCL.1 MAP2K5
DVKPSNMLVNTR
Lys2
-4.198608382
1
uM
QL-XII-47 MWCL.1 MAP2K6
DVKPSNVLINALGQVK
Lys2
5.39398113
1
uM
QL-XII-47 MWCL.1 MP2K7
DVKPSNILLDER
Lys2
-45.5174114
1
uM
QL-XII-47 MWCL.1 MAP3K1
DVKGANLLIDSTGQR
Lys2
9.175244255
1
uM
QL-XII-47 MWCL.1 M3K2
ELAVKQVQFDPDSPETSKEVNALECEIQLLK
Lys1
-0.459368027
1
uM
QL-XII-47 MWCL.1 M3K2,MAP3K3
DIKGANILR
Lys2
17.59521009
1
uM
QL-XII-47 MWCL.1 MAP3K3
ELASKQVQFDPDSPETSKEVSALECEIQLLK
Lys1
-1.791203787
1
uM
QL-XII-47 MWCL.1 MAP3K4
DIKGANIFLTSSGLIK
Lys2
16.84992087
1
uM
QL-XII-47 MWCL.1 MAP3K5
DIKGDNVLINTYSGVLK
Lys2
-9.625870933
1
uM
QL-XII-47 MWCL.1 MARK2,MARK3
DLKAENLLLDADMNIK
Lys2
-11.86915829
1
uM
QL-XII-47 MWCL.1 MARK3
EVAIKIIDKTQLNPTSLQK
Lys1
10.94267365
1
uM
QL-XII-47 MWCL.1 MARK3,MARK4
EVAIKIIDK
Lys1
5.793943076
1
uM
QL-XII-47 MWCL.1 MAST1,MAST2
DLKPDNLLITSMGHIK
Lys2
-89.96758232
1
uM
QL-XII-47 MWCL.1 MAST3
DLKPDNLLITSLGHIK
Lys2
3.312930204
1
uM
QL-XII-47 MWCL.1 MASTL
GAFGKVYLGQK
ATP Loop
-5.128672656
1
uM
QL-XII-47 MWCL.1 MASTL
LYAVKVVK
Lys1
-4.9183009
1
uM
QL-XII-47 MWCL.1 MLK3
DLKSNNILLLQPIESDDMEHK
Lys2
24.61377493
1
uM