QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
QL-XII-47 | MWCL.1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 5.905585783 | 1 | uM |
QL-XII-47 | MWCL.1 | LOK | DLKAGNVLMTLEGDIR | Lys2 | -3.152905014 | 1 | uM |
QL-XII-47 | MWCL.1 | LRRK2 | DLKPHNVLLFTLYPNAAIIAK | Lys2 | 7.098641111 | 1 | uM |
QL-XII-47 | MWCL.1 | LYN | VAVKTLKPGTMSVQAFLEEANLMK | Lys1 | 2.528406343 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP2K1 | IMHRDVKPSNILVNSR | Lys2 | -10.45585154 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | 2.14775294 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP2K3 | DVKPSNVLINK | Lys2 | -11.1285874 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP2K4 | DIKPSNILLDR | Lys2 | -4.661208852 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP2K5 | DVKPSNMLVNTR | Lys2 | -4.198608382 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP2K6 | DVKPSNVLINALGQVK | Lys2 | 5.39398113 | 1 | uM |
QL-XII-47 | MWCL.1 | MP2K7 | DVKPSNILLDER | Lys2 | -45.5174114 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | 9.175244255 | 1 | uM |
QL-XII-47 | MWCL.1 | M3K2 | ELAVKQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -0.459368027 | 1 | uM |
QL-XII-47 | MWCL.1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | 17.59521009 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP3K3 | ELASKQVQFDPDSPETSKEVSALECEIQLLK | Lys1 | -1.791203787 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | 16.84992087 | 1 | uM |
QL-XII-47 | MWCL.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | -9.625870933 | 1 | uM |
QL-XII-47 | MWCL.1 | MARK2,MARK3 | DLKAENLLLDADMNIK | Lys2 | -11.86915829 | 1 | uM |
QL-XII-47 | MWCL.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | 10.94267365 | 1 | uM |
QL-XII-47 | MWCL.1 | MARK3,MARK4 | EVAIKIIDK | Lys1 | 5.793943076 | 1 | uM |
QL-XII-47 | MWCL.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | -89.96758232 | 1 | uM |
QL-XII-47 | MWCL.1 | MAST3 | DLKPDNLLITSLGHIK | Lys2 | 3.312930204 | 1 | uM |
QL-XII-47 | MWCL.1 | MASTL | GAFGKVYLGQK | ATP Loop | -5.128672656 | 1 | uM |
QL-XII-47 | MWCL.1 | MASTL | LYAVKVVK | Lys1 | -4.9183009 | 1 | uM |
QL-XII-47 | MWCL.1 | MLK3 | DLKSNNILLLQPIESDDMEHK | Lys2 | 24.61377493 | 1 | uM |