QL-XII-47 KiNativ -- single dose experiment - Dataset (ID:20205)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-XII-47 | BCWM.1 | LCK | EGAKFPIKWTAPEAINYGTFTIK | Activation Loop | -3.451280562 | 1 | uM |
| QL-XII-47 | BCWM.1 | M3K6 | DIKGDNVLINTFSGLLK | Lys2 | -28.65680338 | 1 | uM |
| QL-XII-47 | BCWM.1 | MARK4 | DLKAENLLLDAEANIK | Lys2 | -5.460937261 | 1 | uM |
| QL-XII-47 | BCWM.1 | MELK | DLKPENLLFDEYHK | Lys2 | -16.2088292 | 1 | uM |
| QL-XII-47 | BCWM.1 | NEK2 | DLKPANVFLDGK | Lys2 | 0.142322043 | 1 | uM |
| QL-XII-47 | BCWM.1 | CDK16 | SKLTDNLVALKEIR | Lys1 | 29.54620403 | 1 | uM |
| QL-XII-47 | BCWM.1 | RSK2 domain1 | DLKPENILLDEEGHIKLTDFGLSKESIDHEK | Lys2 | -55.49739312 | 1 | uM |
| QL-XII-47 | BCWM.1 | STK33 | DLKLENIMVK | Lys2 | 21.08514361 | 1 | uM |
| QL-XII-47 | BCWM.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 0.574708889 | 1 | uM |
| QL-XII-47 | BCWM.1 | Wnk1,Wnk2 | GSFKTVYK | ATP Loop | -23.10912536 | 1 | uM |
| QL-XII-47 | MWCL.1 | BLK | IIDSEYTAQEGAKFPIK | Activation Loop | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | -6.530594283 | 1 | uM |
| QL-XII-47 | MWCL.1 | KCC4 | DLKPENLLYATPAPDAPLK | Lys2 | -26.82702802 | 1 | uM |
| QL-XII-47 | MWCL.1 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 0.240956147 | 1 | uM |
| QL-XII-47 | MWCL.1 | EPHB1 | YLQDDTSDPTYTSSLGGKIPVR | Activation Loop | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 6.167010891 | 1 | uM |
| QL-XII-47 | MWCL.1 | FRK | HEIKLPVK | Activation Loop | 7.187023655 | 1 | uM |
| QL-XII-47 | MWCL.1 | KSR1 | SKNVFYDNGKVVITDFGLFGISGVVR | Activation Loop | -32.14952167 | 1 | uM |
| QL-XII-47 | MWCL.1 | LCK | EGAKFPIKWTAPEAINYGTFTIK | Activation Loop | -28.69047225 | 1 | uM |
| QL-XII-47 | MWCL.1 | M3K6 | DIKGDNVLINTFSGLLK | Lys2 | ND | 1 | uM |
| QL-XII-47 | MWCL.1 | MARK4 | DLKAENLLLDAEANIK | Lys2 | -23.76148008 | 1 | uM |
| QL-XII-47 | MWCL.1 | MELK | DLKPENLLFDEYHK | Lys2 | 7.74246842 | 1 | uM |
| QL-XII-47 | MWCL.1 | NEK2 | DLKPANVFLDGK | Lys2 | -13.95606145 | 1 | uM |
| QL-XII-47 | MWCL.1 | CDK16 | SKLTDNLVALKEIR | Lys1 | 15.03393916 | 1 | uM |
| QL-XII-47 | MWCL.1 | RSK2 domain1 | DLKPENILLDEEGHIKLTDFGLSKESIDHEK | Lys2 | -48.46241013 | 1 | uM |