TG-101348 KINOMEscan - Dataset (ID:20174)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Fedratinib | MP2K4 | 9900.0 | nM |
Fedratinib | RIPK4 | 9800.0 | nM |
Fedratinib | BRAF | 9800.0 | nM |
Fedratinib | MLCK | 9700.0 | nM |
Fedratinib | KPCD3 | 9600.0 | nM |
Fedratinib | DYRK1B | 9500.0 | nM |
Fedratinib | BRAF(V600E) | 9300.0 | nM |
Fedratinib | MINK | 8900.0 | nM |
Fedratinib | CDK9 | 8800.0 | nM |
Fedratinib | CDK15 | 8600.0 | nM |
Fedratinib | TRKC | 8600.0 | nM |
Fedratinib | MET | 8500.0 | nM |
Fedratinib | KPCE | 8100.0 | nM |
Fedratinib | RSK2(Kin.Dom.1-N-terminal) | 8100.0 | nM |
Fedratinib | LATS2 | 8000.0 | nM |
Fedratinib | LIMK2 | 7900.0 | nM |
Fedratinib | RSK3(Kin.Dom.1-N-terminal) | 7700.0 | nM |
Fedratinib | EPHA8 | 7700.0 | nM |
Fedratinib | PIK3CG | 7500.0 | nM |
Fedratinib | MST4 | 7500.0 | nM |
Fedratinib | CDKL5 | 7300.0 | nM |
Fedratinib | MKNK1 | 7300.0 | nM |
Fedratinib | YSK1 | 7200.0 | nM |
Fedratinib | EPHA3 | 7100.0 | nM |
Fedratinib | ADCK3 | 7000.0 | nM |