CI-1033 KINOMEscan-2 - Dataset (ID:20164)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Canertinib | EGFR(T790M) | 0.10 | nM |
Canertinib | EGFR(G719C) | 0.13 | nM |
Canertinib | EGFR(L747-E749del, A750P) | 0.17 | nM |
Canertinib | EGFR | 0.19 | nM |
Canertinib | EGFR(S752-I759del) | 0.19 | nM |
Canertinib | EGFR(G719S) | 0.19 | nM |
Canertinib | EGFR(L861Q) | 0.22 | nM |
Canertinib | EGFR(L858R) | 0.24 | nM |
Canertinib | EGFR(L747-S752del, P753S) | 0.26 | nM |
Canertinib | EGFR(E746-A750del) | 0.26 | nM |
Canertinib | EGFR(L747-T751del,Sins) | 0.26 | nM |
Canertinib | EGFR(L858R,T790M) | 0.28 | nM |
Canertinib | ERBB4 | 6.50 | nM |
Canertinib | ABL1(Q252H)-phosphorylated | 22.00 | nM |
Canertinib | ABL1(E255K)-phosphorylated | 30.00 | nM |
Canertinib | ABL1-phosphorylated | 30.00 | nM |
Canertinib | ABL1(M351T)-phosphorylated | 38.00 | nM |
Canertinib | ABL1(Y253F)-phosphorylated | 42.00 | nM |
Canertinib | BLK | 45.00 | nM |
Canertinib | ABL1(H396P)-nonphosphorylated | 46.00 | nM |
Canertinib | ERBB2 | 56.00 | nM |
Canertinib | ABL1(H396P)-phosphorylated | 57.00 | nM |
Canertinib | MP2K5 | 60.00 | nM |
Canertinib | ABL1(T315I)-phosphorylated | 69.00 | nM |
Canertinib | ABL1(F317L)-phosphorylated | 91.00 | nM |