CI-1033 KINOMEscan-2 - Dataset (ID:20164)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Canertinib | TGFBR1 | 9600.00 | nM |
Canertinib | RIOK1 | 8400.00 | nM |
Canertinib | MAP3K4 | 8400.00 | nM |
Canertinib | TNIK | 8200.00 | nM |
Canertinib | KIT(V559D) | 7900.00 | nM |
Canertinib | KIT(V559D,V654A) | 7900.00 | nM |
Canertinib | KIT | 7800.00 | nM |
Canertinib | ALK | 7700.00 | nM |
Canertinib | VGFR1 | 7500.00 | nM |
Canertinib | PGFRB | 7500.00 | nM |
Canertinib | DRAK2 | 7300.00 | nM |
Canertinib | DMPK | 7000.00 | nM |
Canertinib | SRMS | 6700.00 | nM |
Canertinib | DYRK2 | 6700.00 | nM |
Canertinib | HUNK | 6400.00 | nM |
Canertinib | RSK1(Kin.Dom.2-C-terminal) | 6200.00 | nM |
Canertinib | CSK | 6100.00 | nM |
Canertinib | AXL | 5700.00 | nM |
Canertinib | KIT(L576P) | 5700.00 | nM |
Canertinib | TNNI3K | 5600.00 | nM |
Canertinib | ITK | 5600.00 | nM |
Canertinib | MET | 5600.00 | nM |
Canertinib | JNK3 | 5500.00 | nM |
Canertinib | ERK4 | 5400.00 | nM |
Canertinib | FYN | 5300.00 | nM |