AMG-706 KINOMEscan - Dataset (ID:20150)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Motesanib | KIT(L576P) | 1.3 | nM |
Motesanib | KIT(V559D) | 3.2 | nM |
Motesanib | KIT | 3.7 | nM |
Motesanib | CSF1R | 5.6 | nM |
Motesanib | MLTK | 8.0 | nM |
Motesanib | PGFRB | 9.1 | nM |
Motesanib | FLT4 | 9.7 | nM |
Motesanib | PGFRA | 10.0 | nM |
Motesanib | VGFR1 | 12.0 | nM |
Motesanib | KIT(V559D,T670I) | 13.0 | nM |
Motesanib | RET | 14.0 | nM |
Motesanib | KIT(A829P) | 15.0 | nM |
Motesanib | RET(M918T) | 20.0 | nM |
Motesanib | KIT(V559D,V654A) | 23.0 | nM |
Motesanib | VGFR2 | 26.0 | nM |
Motesanib | FLT3(K663Q) | 54.0 | nM |
Motesanib | FLT3 | 71.0 | nM |
Motesanib | FRK | 99.0 | nM |
Motesanib | LYN | 160.0 | nM |
Motesanib | KIT(D816H) | 180.0 | nM |
Motesanib | YSK4 | 200.0 | nM |
Motesanib | TNNI3K | 220.0 | nM |
Motesanib | DDR1 | 260.0 | nM |
Motesanib | BRAF(V600E) | 280.0 | nM |
Motesanib | CIT | 300.0 | nM |