Metrics other than potency reveal systematic variation in responses to cancer drugs - Dataset (ID:20120)
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Small Molecule | Cell Line | log10[max. dose (M)] | R^2 (goodness of fit) | log10[EC50 (M)] | log10[IC50 (M)] | log10[GI50 (M)] | HillSlope | E_inf | E_max | AUC |
---|---|---|---|---|---|---|---|---|---|---|
Z-Leu-Leu-Norvalinal | HCC1806 | -4.1759 | 0.9667 | -5.9139 | -5.9076 | -5.9880 | 2.5020 | 0.0120 | 0.0120 | 5.6935 |
Z-Leu-Leu-Norvalinal | HCC1937 | -4.1759 | 0.9971 | -6.0099 | -6.0088 | -6.3789 | 3.9990 | 0.0058 | 0.0058 | 5.9138 |
Z-Leu-Leu-Norvalinal | HCC1954 | -4.1759 | 0.9781 | -6.1469 | -6.1454 | -6.2118 | 3.3340 | 0.0072 | 0.0072 | 5.5164 |
Z-Leu-Leu-Norvalinal | HCC202 | -4.1759 | 0.9849 | -6.1109 | -6.0129 | -6.5191 | 2.2650 | 0.1997 | 0.1997 | 6.2528 |
Z-Leu-Leu-Norvalinal | HCC38 | -4.1759 | 0.9811 | -6.1804 | -6.1801 | -6.2592 | 3.9990 | 0.0019 | 0.0019 | 5.5300 |
Z-Leu-Leu-Norvalinal | HCC70 | -4.1759 | 0.9890 | -6.4969 | -6.4931 | -6.8051 | 2.8540 | 0.0120 | 0.0120 | 5.0384 |
Z-Leu-Leu-Norvalinal | Hs 578T | -4.1759 | 0.9799 | -6.1834 | -6.1824 | -6.2573 | 3.7490 | 0.0043 | 0.0043 | 5.7867 |
Z-Leu-Leu-Norvalinal | MB 157 | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN |
Z-Leu-Leu-Norvalinal | MDA-MB-134-VI | -4.1759 | 0.9887 | -6.0569 | -6.0511 | -6.1492 | 3.9990 | 0.0278 | 0.0278 | 5.7423 |
Z-Leu-Leu-Norvalinal | MDA-MB-157 | -4.1759 | 0.9623 | -6.2399 | -6.2359 | -6.4226 | 2.8140 | 0.0148 | 0.0148 | 5.4484 |
Z-Leu-Leu-Norvalinal | MDA-MB-175-VII | -4.1759 | 0.9930 | -5.9949 | -5.9733 | -6.2188 | 2.9240 | 0.0548 | 0.0548 | 6.0043 |
Z-Leu-Leu-Norvalinal | MDA-MB-361 | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN |
Z-Leu-Leu-Norvalinal | MDA-MB-436 | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN |
Z-Leu-Leu-Norvalinal | MDA-MB-453 | -4.1759 | 0.9320 | -6.0599 | -6.0164 | -6.2764 | 1.8470 | 0.0834 | 0.0837 | 5.7261 |
Z-Leu-Leu-Norvalinal | MDA-MB-468 | -4.1759 | 0.9865 | -6.1719 | -6.1694 | -6.2332 | 2.9780 | 0.0119 | 0.0119 | 5.5715 |
Z-Leu-Leu-Norvalinal | T47D | -4.1759 | 0.9856 | -6.0629 | -6.0593 | -6.2439 | 3.9995 | 0.0169 | 0.0169 | 6.0577 |
Z-Leu-Leu-Norvalinal | UACC-812 | -4.1759 | 0.9369 | -5.8419 | -5.7175 | -6.0650 | 1.2500 | 0.1502 | 0.1572 | 6.2475 |
Z-Leu-Leu-Norvalinal | UACC-893 | -4.1759 | 0.9765 | -5.8879 | -5.7936 | -6.0573 | 2.9860 | 0.2385 | 0.2385 | 6.6484 |
Z-Leu-Leu-Norvalinal | ZR-75-1 | -4.1759 | 0.9892 | -5.5389 | -5.4977 | -5.7673 | 2.5590 | 0.1089 | 0.1092 | 6.6666 |
Z-Leu-Leu-Norvalinal | 184B5 | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN |
Z-Leu-Leu-Norvalinal | HCC1187 | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN |
Z-Leu-Leu-Norvalinal | MCF 10A | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN | NaN |
Z-Leu-Leu-Norvalinal | MCF 10F | -4.1759 | 0.9833 | -6.3579 | -6.3502 | -6.6528 | 1.4630 | 0.0129 | 0.0135 | 5.3267 |
Z-Leu-Leu-Norvalinal | SUM1315MO2 | -4.1759 | 0.8595 | -5.9989 | -5.9987 | -6.8638 | 0.9127 | 0.0000 | 0.0212 | 5.7823 |
Z-Leu-Leu-Norvalinal | SUM149PT | -4.1759 | 0.9136 | -6.0154 | -6.0153 | -6.1387 | 2.0675 | 0.0004 | 0.0021 | 5.7558 |