CH5424802 KiNativ -- single dose experiment - Dataset (ID:20105)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
CH5424802 HeLa MAP2K3
MCDFGISGYLVDSVAkTMDAGCKPYMAPER
Activation Loop
5.2
10
uM
CH5424802 HeLa MARK1
EVAVkIIDKTQLNPTSLQK
Lys1
4.7
10
uM
CH5424802 HeLa NUAK1
VVAIkSIR
Lys1
5.2
10
uM
CH5424802 HeLa KPCI
IYAMkVVK
Lys1
13.4
10
uM
CH5424802 HeLa PLK1
EVFAGkIVPK
Lys1
0.5
10
uM
CH5424802 HeLa PRP4
CNILHADIkPDNILVNESK
Lys2
20.9
10
uM
CH5424802 HeLa RSK1 domain1
DLKPENILLDEEGHIkLTDFGLSKEAIDHEK
Lys2
76.9
10
uM
CH5424802 HeLa EGFR
LLGAEEKEYHAEGGkVPIKWMALESILHR
Activation Loop
3.4
10
uM
CH5424802 HeLa EGFR
GLWIPEGEKVKIPVAIkELR
Lys1
-1.4
10
uM
CH5424802 HeLa PLK1
VIHRDLkLGNLFLNEDLEVK
Lys2
-8.9
10
uM