XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-85h HeLa HPK1
DKVSGDLVALkMVK
Lys1
-8.0
10
uM
XMD11-85h HeLa IKKE
SGELVAVkVFNTTSYLRPR
Lys1
-8.5
10
uM
XMD11-85h HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
1.9
10
uM
XMD11-85h HeLa LATS2
VDTHALYAMkTLR
Lys1
-18.0
10
uM
XMD11-85h HeLa LYN
VAVkTLKPGTMSVQAFLEEANLMK
Lys1
4.8
10
uM
XMD11-85h PC-3 M3K2
VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
-37.4
10
uM
XMD11-85h HeLa MAP3K5
DIkGDNVLINTYSGVLK
Lys2
-6.3
10
uM
XMD11-85h HeLa MAPKAPK3
KYAVTDDYQLSkQVLGLGVNGK
ATP Loop
6.0
10
uM
XMD11-85h PC-3 MARK2
EVAVkIIDKTQLNSSSLQK
Lys1
8.8
10
uM
XMD11-85h PC-3 MARK3,MARK4
EVAIkIIDK
Lys1
1.2
10
uM
XMD11-85h HeLa MASTL
LYAVkVVK
Lys1
-2.0
10
uM
XMD11-85h PC-3 MET
DMYDkEYYSVHNK
Activation Loop
27.6
10
uM
XMD11-85h PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
15.0
10
uM
XMD11-85h HeLa p38a
DLkPSNLAVNEDCELK
Lys2
-18.6
10
uM
XMD11-85h PC-3 p38a
DLkPSNLAVNEDCELK
Lys2
9.8
10
uM
XMD11-85h HeLa MK14
QELNkTIWEVPER
Other
-2.2
10
uM
XMD11-85h PC-3 MK14
QELNkTIWEVPER
Other
0.5
10
uM
XMD11-85h HeLa PAN3
VMDPTkILITGK
-10.7
10
uM
XMD11-85h HeLa PEK
DLkPSNIFFTMDDVVK
Lys2
-19.1
10
uM
XMD11-85h PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
17.7
10
uM
XMD11-85h HeLa PIK3CG
KkPLWLEFK
ATP
-25.6
10
uM
XMD11-85h HeLa PKN1
GHFGkVLLSEFRPSGELFAIK
Lys1
33.8
10
uM
XMD11-85h HeLa PLK1
DLkLGNLFLNEDLEVK
Lys2
26.3
10
uM
XMD11-85h PC-3 ROCK1
kLQLELNQER
Other
1.2
10
uM
XMD11-85h PC-3 RON
IQCAIkSLSR
Lys1
10.5
10
uM