XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-85h | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | -8.0 | 10 | uM |
XMD11-85h | HeLa | IKKE | SGELVAVkVFNTTSYLRPR | Lys1 | -8.5 | 10 | uM |
XMD11-85h | HeLa | KSR1,KSR2 | SkNVFYDNGK | Protein Kinase Domain | 1.9 | 10 | uM |
XMD11-85h | HeLa | LATS2 | VDTHALYAMkTLR | Lys1 | -18.0 | 10 | uM |
XMD11-85h | HeLa | LYN | VAVkTLKPGTMSVQAFLEEANLMK | Lys1 | 4.8 | 10 | uM |
XMD11-85h | PC-3 | M3K2 | VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK | Lys1 | -37.4 | 10 | uM |
XMD11-85h | HeLa | MAP3K5 | DIkGDNVLINTYSGVLK | Lys2 | -6.3 | 10 | uM |
XMD11-85h | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | 6.0 | 10 | uM |
XMD11-85h | PC-3 | MARK2 | EVAVkIIDKTQLNSSSLQK | Lys1 | 8.8 | 10 | uM |
XMD11-85h | PC-3 | MARK3,MARK4 | EVAIkIIDK | Lys1 | 1.2 | 10 | uM |
XMD11-85h | HeLa | MASTL | LYAVkVVK | Lys1 | -2.0 | 10 | uM |
XMD11-85h | PC-3 | MET | DMYDkEYYSVHNK | Activation Loop | 27.6 | 10 | uM |
XMD11-85h | PC-3 | MRCKb | NHHVHLYPWSSLDGAEGSFDIkLPETK | Other | 15.0 | 10 | uM |
XMD11-85h | HeLa | p38a | DLkPSNLAVNEDCELK | Lys2 | -18.6 | 10 | uM |
XMD11-85h | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | 9.8 | 10 | uM |
XMD11-85h | HeLa | MK14 | QELNkTIWEVPER | Other | -2.2 | 10 | uM |
XMD11-85h | PC-3 | MK14 | QELNkTIWEVPER | Other | 0.5 | 10 | uM |
XMD11-85h | HeLa | PAN3 | VMDPTkILITGK | -10.7 | 10 | uM | |
XMD11-85h | HeLa | PEK | DLkPSNIFFTMDDVVK | Lys2 | -19.1 | 10 | uM |
XMD11-85h | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 17.7 | 10 | uM |
XMD11-85h | HeLa | PIK3CG | KkPLWLEFK | ATP | -25.6 | 10 | uM |
XMD11-85h | HeLa | PKN1 | GHFGkVLLSEFRPSGELFAIK | Lys1 | 33.8 | 10 | uM |
XMD11-85h | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | 26.3 | 10 | uM |
XMD11-85h | PC-3 | ROCK1 | kLQLELNQER | Other | 1.2 | 10 | uM |
XMD11-85h | PC-3 | RON | IQCAIkSLSR | Lys1 | 10.5 | 10 | uM |