XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-85h HeLa PKD2
DVAVkVIDK
Lys1
-24.7
10
uM
XMD11-85h PC-3 PKD2
DVAVkVIDK
Lys1
28.4
10
uM
XMD11-85h HeLa RIPK3
DLkPSNVLLDPELHVK
Lys2
6.7
10
uM
XMD11-85h HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-23.5
10
uM
XMD11-85h HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
9.0
10
uM
XMD11-85h PC-3 SLK
ETSVLAAAkVIDTK
Lys1
-0.8
10
uM
XMD11-85h HeLa SYK
ISDFGLSkALR
Activation Loop
-11.5
10
uM
XMD11-85h HeLa TLK1
YAAVkIHQLNK
Lys1
4.3
10
uM
XMD11-85h PC-3 TLK1
YAAVkIHQLNK
Lys1
-14.4
10
uM
XMD11-85h HeLa ULK1
DLkPQNILLSNPAGR
Lys2
7.1
10
uM
XMD11-85h HeLa AurB
SHFIVALkVLFK
Lys1
41.7
10
uM
XMD11-85h PC-3 CLK2
LTHTDLkPENILFVNSDYELTYNLEK
Lys2
-1.0
10
uM
XMD11-85h HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
-3.2
10
uM
XMD11-85h HeLa MYO3A,MYO3B
DVkGNNILLTTEGGVK
Lys2
26.4
10
uM
XMD11-85h PC-3 SNRK
DLkPENVVFFEK
Lys2
12.3
10
uM
XMD11-85h HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-11.8
10
uM