XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-85h HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-8.0
10
uM
XMD11-85h PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
4.0
10
uM
XMD11-85h HeLa DMPK
DIkPDNILLDR
Lys2
16.5
10
uM
XMD11-85h PC-3 DNAPK
kGGSWIQEINVAEK
ATP
34.1
10
uM
XMD11-85h HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
-21.2
10
uM
XMD11-85h PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
2.7
10
uM
XMD11-85h HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-28.6
10
uM
XMD11-85h PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
10.7
10
uM
XMD11-85h PC-3 EGFR
IPVAIkELR
Lys1
1.2
10
uM
XMD11-85h PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
-0.5
10
uM
XMD11-85h HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-6.6
10
uM
XMD11-85h PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
11.2
10
uM
XMD11-85h HeLa Erk5
DLkPSNLLVNENCELK
Lys2
-8.8
10
uM
XMD11-85h PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
32.6
10
uM
XMD11-85h HeLa FER
TSVAVkTCKEDLPQELK
Lys1
-20.4
10
uM
XMD11-85h PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
5.0
10
uM
XMD11-85h PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
6.7
10
uM
XMD11-85h HeLa GCK
DTVTSELAAVkIVK
Lys1
-2.7
10
uM
XMD11-85h PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
2.0
10
uM
XMD11-85h HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-7.2
10
uM
XMD11-85h PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
9.4
10
uM
XMD11-85h HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-4.4
10
uM
XMD11-85h HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-46.4
10
uM
XMD11-85h PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
12.1
10
uM
XMD11-85h PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
21.9
10
uM