XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD11-85h | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -8.0 | 10 | uM |
XMD11-85h | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 4.0 | 10 | uM |
XMD11-85h | HeLa | DMPK | DIkPDNILLDR | Lys2 | 16.5 | 10 | uM |
XMD11-85h | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 34.1 | 10 | uM |
XMD11-85h | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | -21.2 | 10 | uM |
XMD11-85h | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 2.7 | 10 | uM |
XMD11-85h | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -28.6 | 10 | uM |
XMD11-85h | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | 10.7 | 10 | uM |
XMD11-85h | PC-3 | EGFR | IPVAIkELR | Lys1 | 1.2 | 10 | uM |
XMD11-85h | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | -0.5 | 10 | uM |
XMD11-85h | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | -6.6 | 10 | uM |
XMD11-85h | PC-3 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 11.2 | 10 | uM |
XMD11-85h | HeLa | Erk5 | DLkPSNLLVNENCELK | Lys2 | -8.8 | 10 | uM |
XMD11-85h | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 32.6 | 10 | uM |
XMD11-85h | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | -20.4 | 10 | uM |
XMD11-85h | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 5.0 | 10 | uM |
XMD11-85h | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 6.7 | 10 | uM |
XMD11-85h | HeLa | GCK | DTVTSELAAVkIVK | Lys1 | -2.7 | 10 | uM |
XMD11-85h | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | 2.0 | 10 | uM |
XMD11-85h | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -7.2 | 10 | uM |
XMD11-85h | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 9.4 | 10 | uM |
XMD11-85h | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -4.4 | 10 | uM |
XMD11-85h | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -46.4 | 10 | uM |
XMD11-85h | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 12.1 | 10 | uM |
XMD11-85h | PC-3 | ILK | ISMADVkFSFQCPGR | Protein Kinase Domain | 21.9 | 10 | uM |