Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 1 of 2: Normalized growth rate inhibition values. - Dataset (ID:20350)
Small Molecules Studied
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HMS LINCS ID | Name | Alternative Names | LINCS ID | Structure Image | PubChem CID |
---|---|---|---|---|---|
11955-1 | SB1-F-22 | (S)-N-(1-benzyl-1H-imidazol-4-yl)-1-cyanopyrrolidine-3-carboxamide | |||
11954-1 | SB1-F-21 | (S)-1-cyano-N-(5-phenylthiazol-2-yl)pyrrolidine-3-carboxamide | |||
11953-1 | PB49673382 | ||||
11952-1 | z-VAE(OMe)-fmk | 5497177 | |||
11951-1 | HY-17542 | PLpro Inhibitor | 44235889 | ||
11950-1 | HBX19818 | HBX 19818; HBX-19818 | 73349008 | ||
11949-1 | USP7-IN-1 | 71278663 | |||
11948-1 | ML-323 | ML323; ML 323 | 60167849 | ||
11947-1 | HY-50736 | DUBs-IN-1 | 16065490 | ||
11946-1 | HY-50737A | DUBs-IN-2 | 16065491 | ||
11945-1 | 1247825-37-1 | 4-cyano-5-(3,5-dichloropyridin-4-yl)sulfanyl-N-(4-methylsulfonylphenyl)thiophene-2-carboxamide; USP7/USP47 inhibitor | 51031028 | ||
11943-1 | SJB2-043 | 2-Phenylbenzo[f][1,3]benzoxazole-4,9-dione | 509070 | ||
11942-1 | HY-17541A | Cysteine Protease inhibitor hydrochloride | |||
10562-1 | Vialinin A | Terrestrin A | 11563133 | ||
10561-1 | Spautin-1 | Spautin 1 | 51037431 | ||
10560-1 | IU1 | IU-1 | 675434 | ||
10559-1 | SJB3-019A | 78358325 | |||
10558-1 | Degrasyn | WP 1130; WP1130; WP-1130 | 11222830 | ||
10556-1 | Doxycycline | Doxytetracycline; Monodox; Oracea; Vibramycin | 54671203 | ||
10554-1 | HBX 41108 | 16065773 | |||
10552-1 | Sepantronium | YM155 | 10126189 | ||
10551-1 | MI-2 | MI 2; MALT1 inhibitor | 45942672 | ||
10550-1 | GW7647 | GW 7647; GW-7647; GW647 | 3392731 | ||
10549-1 | Pimozide | McN-JR-6238; Neoperidole; Opiran; Orap; Pimozidum | 16362 | ||
10548-1 | 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one | STK854993 | 2913480 |