Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 1 of 2: Normalized growth rate inhibition values. - Dataset (ID:20350)

Small Molecules Studied

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  • 1 to 25 of 32 Small Molecules
HMS LINCS ID Name Alternative Names LINCS ID Structure Image PubChem CID
10552-1 Sepantronium
YM155
10126189
10558-1 Degrasyn
WP 1130; WP1130; WP-1130
11222830
10562-1 Vialinin A
Terrestrin A
11563133
11947-1 HY-50736
DUBs-IN-1
16065490
11946-1 HY-50737A
DUBs-IN-2
16065491
10554-1 HBX 41108 16065773
10549-1 Pimozide
McN-JR-6238; Neoperidole; Opiran; Orap; Pimozidum
16362
10265-2 Pevonedistat
MLN 4924; MLN-4924; MLN4924
LSM-6263 16720766
10545-1 LDN57444
LDN-57444; Ubiquitin Thiolesterase L1 Inhibitor; UCH-L1 Inhibitor
24906255
10548-1 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one
STK854993
2913480
10550-1 GW7647
GW 7647; GW-7647; GW647
3392731
10479-2 Mitoxantrone
CL 232325; CL-232325; DHAQ; Novantron; Novantrone
LSM-2481 4212
11951-1 HY-17542
PLpro Inhibitor
44235889
10551-1 MI-2
MI 2; MALT1 inhibitor
45942672
10546-1 P22077
P 22077
46931953
11943-1 SJB2-043
2-Phenylbenzo[f][1,3]benzoxazole-4,9-dione
509070
11945-1 1247825-37-1
4-cyano-5-(3,5-dichloropyridin-4-yl)sulfanyl-N-(4-methylsulfonylphenyl)thiophene-2-carboxamide; USP7/USP47 inhibitor
51031028
10561-1 Spautin-1
Spautin 1
51037431
10543-1 b-AP15 5351435
10556-1 Doxycycline
Doxytetracycline; Monodox; Oracea; Vibramycin
54671203
11952-1 z-VAE(OMe)-fmk 5497177
10547-1 Trifluoperazine
Eskazine; Flurazine; Jatroneural; Modalina; Stelazine; Terfluzine; Trifluoperazina; Trifluoroperazine; Trifluperazine; Triflurin; Triftazin; Triperazine
5566
11948-1 ML-323
ML323; ML 323
60167849
10560-1 IU1
IU-1
675434
11949-1 USP7-IN-1 71278663
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  • 1 to 25 of 32 Small Molecules