Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 1 of 2: Normalized growth rate inhibition values. - Dataset (ID:20350)
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Cell | Small Molecule | Small Mol Concentration (uM) | Mean Normalized Growth Rate Inhibition (GR) Value | Increased Fraction Dead |
---|---|---|---|---|
Hs 578T | SJB3-019A | 0.009992797 | 1.1172 | -0.01104 |
MDA-MB-134-VI | Doxycycline | 3.16 | 0.6200 | -0.01100 |
PDX1258 | HBX19818 | 0.009992797 | 0.9600 | -0.01099 |
MDA-MB-134-VI | z-VAE(OMe)-fmk | 0.316 | 0.9482 | -0.01098 |
MDA-MB-361 | IU1 | 3.16 | 1.0450 | -0.01092 |
HCC1500 | IU1 | 0.999279741 | 1.0544 | -0.01090 |
PDX1258 | Spautin-1 | 9.992797406 | 0.8079 | -0.01087 |
PDXHCI002 | SB1-F-21 | 0.0316 | 1.1432 | -0.01086 |
HCC1954 | ML-323 | 0.0316 | 0.9641 | -0.01080 |
Hs 578T | MI-2 | 0.0316 | 1.0217 | -0.01079 |
PDX1328 | HY-17542 | 0.0316 | 1.1924 | -0.01075 |
HCC1937 | Degrasyn | 0.316 | 1.0944 | -0.01074 |
MDA-MB-361 | z-VAE(OMe)-fmk | 0.999279741 | 1.0995 | -0.01073 |
MDA-MB-134-VI | LDN57444 | 0.099927974 | 0.7851 | -0.01071 |
MDA-MB-361 | LDN57444 | 0.999279741 | 1.1609 | -0.01071 |
PDX1258 | STK547622 | 50.0 | 1.0771 | -0.01070 |
BT-549 | Doxycycline | 0.999279741 | 0.9946 | -0.01065 |
PDX1328 | SB1-F-21 | 0.099927974 | 1.0722 | -0.01065 |
PDX1328 | SJB2-043 | 0.0316 | 1.1810 | -0.01065 |
SK-BR-3 | STK547622 | 50.0 | 1.0316 | -0.01065 |
HCC1428 | SJB3-019A | 0.099927974 | 0.9068 | -0.01061 |
BT-20 | IU1 | 0.099927974 | 1.0162 | -0.01061 |
BT-20 | HY-17542 | 0.316 | 1.0486 | -0.01058 |
Hs 578T | USP7-IN-1 | 0.0316 | 1.0637 | -0.01056 |
PDX1328 | z-VAE(OMe)-fmk | 9.992797406 | 0.9702 | -0.01055 |