Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)

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Cell Small Molecule Small Mol Concentration (uM) Primary Target Pathway Mean Normalized Growth Rate Inhibition Value Increased Fraction Dead
BT-20 Ceritinib
0.0031623
ALK
RTK
1.0478 -0.00217
BT-20 Ceritinib
0.01
ALK
RTK
1.0693 -0.00162
BT-20 Ceritinib
0.1
ALK
RTK
1.0073 0.00247
BT-20 Ceritinib
0.31623
ALK
RTK
0.9637 0.00976
BT-20 Abemaciclib
0.001
CDK4/6
Cell cycle
0.9370 -0.00149
BT-20 Abemaciclib
0.0031623
CDK4/6
Cell cycle
0.8833 -0.00527
BT-20 Abemaciclib
0.031623
CDK4/6
Cell cycle
0.4936 -0.00426
BT-20 Abemaciclib
0.1
CDK4/6
Cell cycle
0.3565 0.00950
BT-20 Abemaciclib
3.1623
CDK4/6
Cell cycle
0.1622 0.01068
BT-20 Abemaciclib
10.0
CDK4/6
Cell cycle
-0.2160 0.37259
BT-20 Palbociclib
0.001
CDK4/6
Cell cycle
1.0987 -0.00539
BT-20 Palbociclib
0.0031623
CDK4/6
Cell cycle
0.9966 0.00011
BT-20 Palbociclib
0.31623
CDK4/6
Cell cycle
0.2359 0.04751
BT-20 Palbociclib
1.0
CDK4/6
Cell cycle
0.2044 0.04646
BT-20 AZD7762
0.001
CHK1/2
Cell cycle
1.1198 -0.00253
BT-20 AZD7762
0.0031623
CHK1/2
Cell cycle
1.2431 -0.00726
BT-20 AZD7762
0.1
CHK1/2
Cell cycle
1.1714 0.04490
BT-20 AZD7762
0.31623
CHK1/2
Cell cycle
0.9454 0.07692
BT-20 AZD7762
3.1623
CHK1/2
Cell cycle
-0.1525 0.50057
BT-20 AZD7762
10.0
CHK1/2
Cell cycle
-0.5785 0.71162
BT-20 Volasertib
0.01
PLK
Cell cycle
0.0133 0.34529
BT-20 Volasertib
0.031623
PLK
Cell cycle
-0.4356 0.63889
BT-20 Volasertib
0.31623
PLK
Cell cycle
-0.5339 0.71936
BT-20 Neratinib
0.031623
EGFR/HER2
RTK
0.9331 0.02815
BT-20 Neratinib
0.01
EGFR/HER2
RTK
0.9924 0.00434