Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
BT-20 | Ceritinib | 0.0031623 | ALK | RTK | 1.0478 | -0.00217 |
BT-20 | Ceritinib | 0.01 | ALK | RTK | 1.0693 | -0.00162 |
BT-20 | Ceritinib | 0.1 | ALK | RTK | 1.0073 | 0.00247 |
BT-20 | Ceritinib | 0.31623 | ALK | RTK | 0.9637 | 0.00976 |
BT-20 | Abemaciclib | 0.001 | CDK4/6 | Cell cycle | 0.9370 | -0.00149 |
BT-20 | Abemaciclib | 0.0031623 | CDK4/6 | Cell cycle | 0.8833 | -0.00527 |
BT-20 | Abemaciclib | 0.031623 | CDK4/6 | Cell cycle | 0.4936 | -0.00426 |
BT-20 | Abemaciclib | 0.1 | CDK4/6 | Cell cycle | 0.3565 | 0.00950 |
BT-20 | Abemaciclib | 3.1623 | CDK4/6 | Cell cycle | 0.1622 | 0.01068 |
BT-20 | Abemaciclib | 10.0 | CDK4/6 | Cell cycle | -0.2160 | 0.37259 |
BT-20 | Palbociclib | 0.001 | CDK4/6 | Cell cycle | 1.0987 | -0.00539 |
BT-20 | Palbociclib | 0.0031623 | CDK4/6 | Cell cycle | 0.9966 | 0.00011 |
BT-20 | Palbociclib | 0.31623 | CDK4/6 | Cell cycle | 0.2359 | 0.04751 |
BT-20 | Palbociclib | 1.0 | CDK4/6 | Cell cycle | 0.2044 | 0.04646 |
BT-20 | AZD7762 | 0.001 | CHK1/2 | Cell cycle | 1.1198 | -0.00253 |
BT-20 | AZD7762 | 0.0031623 | CHK1/2 | Cell cycle | 1.2431 | -0.00726 |
BT-20 | AZD7762 | 0.1 | CHK1/2 | Cell cycle | 1.1714 | 0.04490 |
BT-20 | AZD7762 | 0.31623 | CHK1/2 | Cell cycle | 0.9454 | 0.07692 |
BT-20 | AZD7762 | 3.1623 | CHK1/2 | Cell cycle | -0.1525 | 0.50057 |
BT-20 | AZD7762 | 10.0 | CHK1/2 | Cell cycle | -0.5785 | 0.71162 |
BT-20 | Volasertib | 0.01 | PLK | Cell cycle | 0.0133 | 0.34529 |
BT-20 | Volasertib | 0.031623 | PLK | Cell cycle | -0.4356 | 0.63889 |
BT-20 | Volasertib | 0.31623 | PLK | Cell cycle | -0.5339 | 0.71936 |
BT-20 | Neratinib | 0.031623 | EGFR/HER2 | RTK | 0.9331 | 0.02815 |
BT-20 | Neratinib | 0.01 | EGFR/HER2 | RTK | 0.9924 | 0.00434 |