Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
BT-549 | Palbociclib | 1.0 | CDK4/6 | Cell cycle | 1.0826 | -0.00648 |
BT-549 | AZD7762 | 0.001 | CHK1/2 | Cell cycle | 1.1190 | -0.00579 |
BT-549 | AZD7762 | 0.1 | CHK1/2 | Cell cycle | 0.1731 | 0.28658 |
BT-549 | Palbociclib | 0.01 | CDK4/6 | Cell cycle | 1.0649 | 0.00372 |
BT-549 | Palbociclib | 0.0031623 | CDK4/6 | Cell cycle | 1.0202 | -0.00027 |
BT-549 | Palbociclib | 0.031623 | CDK4/6 | Cell cycle | 1.0582 | -0.00203 |
BT-549 | Palbociclib | 0.00031623 | CDK4/6 | Cell cycle | 1.0163 | 0.00360 |
BT-549 | Abemaciclib | 10.0 | CDK4/6 | Cell cycle | 0.0333 | 0.15095 |
BT-549 | Palbociclib | 0.001 | CDK4/6 | Cell cycle | 1.0331 | 0.00886 |
BT-549 | Palbociclib | 0.1 | CDK4/6 | Cell cycle | 1.0491 | 0.00209 |
BT-549 | Abemaciclib | 1.0 | CDK4/6 | Cell cycle | 0.8898 | 0.00509 |
BT-549 | Abemaciclib | 3.1623 | CDK4/6 | Cell cycle | 0.5941 | 0.02941 |
BT-549 | Palbociclib | 0.31623 | CDK4/6 | Cell cycle | 1.0356 | -0.00357 |
BT-549 | AZD7762 | 0.31623 | CHK1/2 | Cell cycle | -0.0478 | 0.29963 |
BT-549 | AZD7762 | 1.0 | CHK1/2 | Cell cycle | -0.1763 | 0.38276 |
BT-549 | Abemaciclib | 0.31623 | CDK4/6 | Cell cycle | 0.9772 | -0.01089 |
BT-549 | Abemaciclib | 0.1 | CDK4/6 | Cell cycle | 0.9609 | 0.00055 |
BT-549 | Abemaciclib | 0.031623 | CDK4/6 | Cell cycle | 0.9941 | -0.00435 |
BT-549 | Abemaciclib | 0.01 | CDK4/6 | Cell cycle | 1.0191 | 0.00387 |
BT-549 | Abemaciclib | 0.0031623 | CDK4/6 | Cell cycle | 1.0379 | -0.00284 |
BT-549 | Abemaciclib | 0.001 | CDK4/6 | Cell cycle | 0.9933 | -0.00259 |
BT-549 | AZD7762 | 3.1623 | CHK1/2 | Cell cycle | -0.2965 | 0.40328 |
BT-549 | Etoposide | 10.0 | Topo II | Chemotherapy | -0.1948 | 0.35550 |
BT-549 | Everolimus | 0.01 | mTOR1 | PI3K/mTOR | 0.5609 | 0.04190 |
BT-549 | Everolimus | 0.0031623 | mTOR1 | PI3K/mTOR | 0.5766 | 0.01630 |