Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
A-375 Vemurafenib Veliparib 1.0000 0.5333
uM
48
hr
2 2518 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 186.55 NGFR rabbit IgG(H+L) / donkey NGFR 195.58
A375-B1-rep2
C2
A-375 Vemurafenib UNC669 1.0000 0.5333
uM
48
hr
2 2288 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 162.78 NGFR rabbit IgG(H+L) / donkey NGFR 184.93
A375-B1-rep2
B8
A-375 Vemurafenib PFI-1 1.0000 0.5333
uM
48
hr
2 2340 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 155.42 NGFR rabbit IgG(H+L) / donkey NGFR 204.08
A375-B1-rep2
B7
A-375 Vemurafenib GSK-J1 1.0000 0.5333
uM
48
hr
2 2749 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 153.27 NGFR rabbit IgG(H+L) / donkey NGFR 180.25
A375-B1-rep2
B6
A-375 Vemurafenib MC1568 1.0000 0.5333
uM
48
hr
2 2064 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 299.54 NGFR rabbit IgG(H+L) / donkey NGFR 157.98
A375-B1-rep2
G4
A-375 Vemurafenib Rocilinostat 1.0000 0.5333
uM
48
hr
2 2904 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 288.39 NGFR rabbit IgG(H+L) / donkey NGFR 128.70
A375-B1-rep2
B5
A-375 Vemurafenib CTB 1.0000 0.5333
uM
48
hr
2 2694 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 159.97 NGFR rabbit IgG(H+L) / donkey NGFR 139.51
A375-B1-rep2
B4
A-375 Vemurafenib Iniparib 1.0000 0.5333
uM
48
hr
2 2392 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 155.20 NGFR rabbit IgG(H+L) / donkey NGFR 165.74
A375-B1-rep2
B3
A-375 Vemurafenib 1.0000
uM
48
hr
2 1429 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 185.39 NGFR rabbit IgG(H+L) / donkey NGFR 144.00
A375-B1-rep2
H10
A-375 Vemurafenib Olaparib 1.0000 0.5333
uM
48
hr
2 2162 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 173.14 NGFR rabbit IgG(H+L) / donkey NGFR 197.62
A375-B1-rep2
B2
A-375 Vemurafenib 1.0000
uM
48
hr
2 1958 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 162.65 NGFR rabbit IgG(H+L) / donkey NGFR 176.09
A375-B1-rep2
A9
A-375 Vemurafenib 1.0000
uM
48
hr
2 1975 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 186.12 NGFR rabbit IgG(H+L) / donkey NGFR 191.67
A375-B1-rep2
A7
A-375 Vemurafenib 1.0000
uM
48
hr
2 1303 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 204.72 NGFR rabbit IgG(H+L) / donkey NGFR 152.30
A375-B1-rep2
H4
A-375 Vemurafenib 1.0000
uM
48
hr
2 2302 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 198.28 NGFR rabbit IgG(H+L) / donkey NGFR 170.70
A375-B1-rep2
A6
A-375 Vemurafenib 1.0000
uM
48
hr
2 1701 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 187.13 NGFR rabbit IgG(H+L) / donkey NGFR 188.45
A375-B1-rep2
A5
A-375 Vemurafenib 1.0000
uM
48
hr
2 2208 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 193.23 NGFR rabbit IgG(H+L) / donkey NGFR 197.15
A375-B1-rep2
A4
A-375 Vemurafenib 1.0000
uM
48
hr
2 2312 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 193.78 NGFR rabbit IgG(H+L) / donkey NGFR 179.41
A375-B1-rep2
A3
A-375 Vemurafenib 1.0000
uM
48
hr
2 2108 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 195.39 NGFR rabbit IgG(H+L) / donkey NGFR 201.04
A375-B1-rep2
A2
A-375 Vemurafenib 1.0000
uM
48
hr
2 1490 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 206.53 NGFR rabbit IgG(H+L) / donkey NGFR 194.20
A375-B1-rep2
A11
A-375 Vemurafenib 1.0000
uM
48
hr
1 2345 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 172.31 NGFR rabbit IgG(H+L) / donkey NGFR 193.43
A375-B2-rep1
A5
A-375 Vemurafenib 1.0000
uM
48
hr
1 2754 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 179.51 NGFR rabbit IgG(H+L) / donkey NGFR 205.98
A375-B2-rep1
A4
A-375 Vemurafenib 1.0000
uM
48
hr
1 2443 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 184.77 NGFR rabbit IgG(H+L) / donkey NGFR 168.94
A375-B2-rep1
A3
A-375 Vemurafenib 1.0000
uM
48
hr
1 2478 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 193.11 NGFR rabbit IgG(H+L) / donkey NGFR 175.65
A375-B2-rep1
A2
A-375 Vemurafenib 1.0000
uM
48
hr
1 2280 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 223.55 NGFR rabbit IgG(H+L) / donkey NGFR 187.85
A375-B2-rep1
A11
A-375 Vemurafenib 1.0000
uM
48
hr
1 2268 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 202.77 NGFR rabbit IgG(H+L) / donkey NGFR 187.51
A375-B2-rep1
A10