Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
A-375 Vemurafenib MC1568 1.0000 0.1067
uM
48
hr
1 2089 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 205.11 NGFR rabbit IgG(H+L) / donkey NGFR 176.85
A375-B2-rep1
G4
A-375 Vemurafenib Ischemin 1.0000 0.1067
uM
48
hr
1 1998 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 186.72 NGFR rabbit IgG(H+L) / donkey NGFR 161.90
A375-B2-rep1
G7
A-375 Vemurafenib Olaparib 1.0000 0.1067
uM
48
hr
2 2141 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 172.10 NGFR rabbit IgG(H+L) / donkey NGFR 172.84
A375-B2-rep2
B2
A-375 Vemurafenib CTB 1.0000 0.1067
uM
48
hr
2 2227 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 169.07 NGFR rabbit IgG(H+L) / donkey NGFR 150.81
A375-B2-rep2
B4
A-375 Vemurafenib Rocilinostat 1.0000 0.1067
uM
48
hr
2 2628 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 191.87 NGFR rabbit IgG(H+L) / donkey NGFR 176.86
A375-B2-rep2
B5
A-375 Vemurafenib Olaparib 1.0000 0.1067
uM
48
hr
1 2585 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 174.02 NGFR rabbit IgG(H+L) / donkey NGFR 185.93
A375-B2-rep1
B2
A-375 Vemurafenib Iniparib 1.0000 0.1067
uM
48
hr
1 2591 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 168.78 NGFR rabbit IgG(H+L) / donkey NGFR 183.97
A375-B2-rep1
B3
A-375 Vemurafenib Rocilinostat 1.0000 0.1067
uM
48
hr
1 2966 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 230.12 NGFR rabbit IgG(H+L) / donkey NGFR 190.47
A375-B2-rep1
B5
A-375 Vemurafenib GSK-J1 1.0000 0.1067
uM
48
hr
1 2690 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 178.62 NGFR rabbit IgG(H+L) / donkey NGFR 187.40
A375-B2-rep1
B6
A-375 Vemurafenib Veliparib 1.0000 0.1067
uM
48
hr
1 2645 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 157.72 NGFR rabbit IgG(H+L) / donkey NGFR 170.56
A375-B2-rep1
C2
A-375 Vemurafenib Rucaparib 1.0000 0.1067
uM
48
hr
1 2454 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 162.10 NGFR rabbit IgG(H+L) / donkey NGFR 185.00
A375-B2-rep1
C3
A-375 Vemurafenib Selisistat 1.0000 0.1067
uM
48
hr
1 3138 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 229.27 NGFR rabbit IgG(H+L) / donkey NGFR 239.03
A375-B2-rep1
C5
A-375 Vemurafenib GSK-J2 1.0000 0.1067
uM
48
hr
1 3266 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 196.57 NGFR rabbit IgG(H+L) / donkey NGFR 202.00
A375-B2-rep1
C6
A-375 Vemurafenib JW55 1.0000 0.1067
uM
48
hr
1 2745 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 171.36 NGFR rabbit IgG(H+L) / donkey NGFR 189.88
A375-B2-rep1
D3
A-375 Vemurafenib Entinostat 1.0000 0.1067
uM
48
hr
1 3329 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 267.58 NGFR rabbit IgG(H+L) / donkey NGFR 296.57
A375-B2-rep1
D4
A-375 Vemurafenib GSK-J4 1.0000 0.1067
uM
48
hr
1 3386 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 161.57 NGFR rabbit IgG(H+L) / donkey NGFR 228.63
A375-B2-rep1
D6
A-375 Vemurafenib (-)-JQ1 1.0000 0.1067
uM
48
hr
1 3182 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 171.84 NGFR rabbit IgG(H+L) / donkey NGFR 203.99
A375-B2-rep1
D7
A-375 Vemurafenib C646 1.0000 0.1067
uM
48
hr
1 2669 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 187.99 NGFR rabbit IgG(H+L) / donkey NGFR 202.06
A375-B2-rep1
E3
A-375 Vemurafenib Mocetinostat 1.0000 0.1067
uM
48
hr
1 2929 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 280.55 NGFR rabbit IgG(H+L) / donkey NGFR 517.04
A375-B2-rep1
E4
A-375 Vemurafenib Daminozide 1.0000 0.1067
uM
48
hr
1 3275 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 183.42 NGFR rabbit IgG(H+L) / donkey NGFR 211.84
A375-B2-rep1
E6
A-375 Vemurafenib I-BET 1.0000 0.1067
uM
48
hr
1 3036 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 143.71 NGFR rabbit IgG(H+L) / donkey NGFR 197.93
A375-B2-rep1
E7
A-375 Vemurafenib BIX-01294 1.0000 0.1067
uM
48
hr
1 2703 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 173.26 NGFR rabbit IgG(H+L) / donkey NGFR 174.07
A375-B2-rep1
F5
A-375 Vemurafenib Methylstat 1.0000 0.1067
uM
48
hr
1 2624 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 155.41 NGFR rabbit IgG(H+L) / donkey NGFR 164.98
A375-B2-rep1
F6
A-375 Vemurafenib Rucaparib 1.0000 0.1067
uM
48
hr
2 2239 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 153.46 NGFR rabbit IgG(H+L) / donkey NGFR 159.08
A375-B2-rep2
C3
A-375 Vemurafenib Veliparib 1.0000 0.1067
uM
48
hr
2 2173 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 161.93 NGFR rabbit IgG(H+L) / donkey NGFR 165.85
A375-B2-rep2
C2