Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
A-375 Vemurafenib Tranylcypromine 1.0000 0.5333
uM
48
hr
2 1765 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 166.51 NGFR rabbit IgG(H+L) / donkey NGFR 168.79
A375-B1-rep2
G6
A-375 Vemurafenib UNC0638 1.0000 0.5333
uM
48
hr
2 1689 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 178.69 NGFR rabbit IgG(H+L) / donkey NGFR 113.11
A375-B1-rep2
G5
COLO 858 Vemurafenib MC1568 0.3160 0.5333
uM
48
hr
2 1098 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 323.03 NGFR rabbit IgG(H+L) / donkey NGFR 124.26
Colo858-B1-rep2
G4
A-375 Vemurafenib MC1568 1.0000 0.5333
uM
48
hr
2 2064 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 299.54 NGFR rabbit IgG(H+L) / donkey NGFR 157.98
A375-B1-rep2
G4
A-375 Vemurafenib Anacardic acid 1.0000 0.5333
uM
48
hr
2 1745 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 183.73 NGFR rabbit IgG(H+L) / donkey NGFR 158.90
A375-B1-rep2
G3
A-375 Vemurafenib RG-108 1.0000 0.5333
uM
48
hr
2 1758 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 186.76 NGFR rabbit IgG(H+L) / donkey NGFR 147.11
A375-B1-rep2
G2
A-375 Vemurafenib CX-5461 1.0000 0.5333
uM
48
hr
2 1227 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 123.06 NGFR rabbit IgG(H+L) / donkey NGFR 136.57
A375-B1-rep2
F8
COLO 858 Vemurafenib RG-108 0.3160 0.5333
uM
48
hr
2 1025 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 269.93 NGFR rabbit IgG(H+L) / donkey NGFR 130.25
Colo858-B1-rep2
G2
A-375 Vemurafenib I-BET151 1.0000 0.5333
uM
48
hr
2 2401 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 153.82 NGFR rabbit IgG(H+L) / donkey NGFR 109.14
A375-B1-rep2
F7
A-375 Vemurafenib Methylstat 1.0000 0.5333
uM
48
hr
2 2362 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 141.85 NGFR rabbit IgG(H+L) / donkey NGFR 141.45
A375-B1-rep2
F6
A-375 Vemurafenib BIX-01294 1.0000 0.5333
uM
48
hr
2 2173 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 148.24 NGFR rabbit IgG(H+L) / donkey NGFR 105.39
A375-B1-rep2
F5
A-375 Vemurafenib Pracinostat 1.0000 0.5333
uM
48
hr
2 2095 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 492.96 NGFR rabbit IgG(H+L) / donkey NGFR 61.23
A375-B1-rep2
F4
COLO 858 Vemurafenib Anacardic acid 0.3160 0.5333
uM
48
hr
2 926 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 272.48 NGFR rabbit IgG(H+L) / donkey NGFR 124.30
Colo858-B1-rep2
G3
COLO 858 Vemurafenib UNC0638 0.3160 0.5333
uM
48
hr
2 1278 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 262.32 NGFR rabbit IgG(H+L) / donkey NGFR 196.87
Colo858-B1-rep2
G5
A-375 Vemurafenib Garcinol 1.0000 0.5333
uM
48
hr
2 2319 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 196.18 NGFR rabbit IgG(H+L) / donkey NGFR 178.69
A375-B1-rep2
F3
A-375 Vemurafenib Decitabine 1.0000 0.5333
uM
48
hr
2 2061 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 195.89 NGFR rabbit IgG(H+L) / donkey NGFR 175.61
A375-B1-rep2
F2
COLO 858 Vemurafenib Pracinostat 0.3160 0.5333
uM
48
hr
2 326 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 166.82 NGFR rabbit IgG(H+L) / donkey NGFR 26.66
Colo858-B1-rep2
F4
A-375 Vemurafenib Epigallocatechin gallate 1.0000 0.5333
uM
48
hr
2 2866 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 196.38 NGFR rabbit IgG(H+L) / donkey NGFR 183.28
A375-B1-rep2
E8
A-375 Vemurafenib I-BET 1.0000 0.5333
uM
48
hr
2 2710 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 145.52 NGFR rabbit IgG(H+L) / donkey NGFR 139.02
A375-B1-rep2
E7
COLO 858 Vemurafenib BIX-01294 0.3160 0.5333
uM
48
hr
2 1928 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 358.98 NGFR rabbit IgG(H+L) / donkey NGFR 120.70
Colo858-B1-rep2
F5
A-375 Vemurafenib Daminozide 1.0000 0.5333
uM
48
hr
2 3093 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 188.94 NGFR rabbit IgG(H+L) / donkey NGFR 179.22
A375-B1-rep2
E6
A-375 Vemurafenib Resveratrol 1.0000 0.5333
uM
48
hr
2 2798 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 177.44 NGFR rabbit IgG(H+L) / donkey NGFR 162.07
A375-B1-rep2
E5
COLO 858 Vemurafenib Decitabine 0.3160 0.5333
uM
48
hr
2 1367 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 214.98 NGFR rabbit IgG(H+L) / donkey NGFR 173.73
Colo858-B1-rep2
F2
A-375 Vemurafenib Mocetinostat 1.0000 0.5333
uM
48
hr
2 2584 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 288.63 NGFR rabbit IgG(H+L) / donkey NGFR 378.86
A375-B1-rep2
E4
A-375 Vemurafenib C646 1.0000 0.5333
uM
48
hr
2 2684 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 170.48 NGFR rabbit IgG(H+L) / donkey NGFR 184.36
A375-B1-rep2
E3