Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
WM-115 Vemurafenib Epigallocatechin gallate 1.0000 0.1067
uM
48
hr
2 1519 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 126.36 NGFR rabbit IgG(H+L) / donkey NGFR 1180.29
WM115-B2-rep2
E8
WM-115 Vemurafenib Pracinostat 1.0000 0.1067
uM
48
hr
2 1651 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 118.63 NGFR rabbit IgG(H+L) / donkey NGFR 885.63
WM115-B2-rep2
F4
WM-115 Vemurafenib BIX-01294 1.0000 0.1067
uM
48
hr
2 1551 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 158.43 NGFR rabbit IgG(H+L) / donkey NGFR 1178.42
WM115-B2-rep2
F5
WM-115 Vemurafenib I-BET151 1.0000 0.1067
uM
48
hr
2 1356 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 127.15 NGFR rabbit IgG(H+L) / donkey NGFR 855.29
WM115-B2-rep2
F7
WM-115 Vemurafenib CX-5461 1.0000 0.1067
uM
48
hr
2 1332 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 124.12 NGFR rabbit IgG(H+L) / donkey NGFR 1219.65
WM115-B2-rep2
F8
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1100 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 149.13 NGFR rabbit IgG(H+L) / donkey NGFR 1179.05
WM115-B2-rep2
A10
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1179 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 152.88 NGFR rabbit IgG(H+L) / donkey NGFR 1171.65
WM115-B2-rep2
A11
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1434 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 159.89 NGFR rabbit IgG(H+L) / donkey NGFR 1166.16
WM115-B2-rep2
A3
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1183 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 156.49 NGFR rabbit IgG(H+L) / donkey NGFR 1100.47
WM115-B2-rep2
A4
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1123 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 140.11 NGFR rabbit IgG(H+L) / donkey NGFR 1122.60
WM115-B2-rep2
A7
WM-115 Vemurafenib 1.0000
uM
48
hr
2 956 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 128.27 NGFR rabbit IgG(H+L) / donkey NGFR 1161.55
WM115-B2-rep2
A8
WM-115 Vemurafenib Olaparib 1.0000 0.1067
uM
48
hr
2 1291 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 154.34 NGFR rabbit IgG(H+L) / donkey NGFR 1162.67
WM115-B2-rep2
B2
WM-115 Vemurafenib Iniparib 1.0000 0.1067
uM
48
hr
2 1353 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 144.10 NGFR rabbit IgG(H+L) / donkey NGFR 1083.77
WM115-B2-rep2
B3
WM-115 Vemurafenib PFI-1 1.0000 0.1067
uM
48
hr
2 1186 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 141.71 NGFR rabbit IgG(H+L) / donkey NGFR 1098.16
WM115-B2-rep2
B7
WM-115 Vemurafenib UNC669 1.0000 0.1067
uM
48
hr
2 1142 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 138.65 NGFR rabbit IgG(H+L) / donkey NGFR 1180.01
WM115-B2-rep2
B8
WM-115 Vemurafenib Rucaparib 1.0000 0.1067
uM
48
hr
2 1286 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 135.71 NGFR rabbit IgG(H+L) / donkey NGFR 1110.95
WM115-B2-rep2
C3
WM-115 Vemurafenib Belinostat 1.0000 0.1067
uM
48
hr
2 1389 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 130.46 NGFR rabbit IgG(H+L) / donkey NGFR 499.87
WM115-B2-rep2
C4
WM-115 Vemurafenib (+)-JQ1 1.0000 0.1067
uM
48
hr
2 1160 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 129.96 NGFR rabbit IgG(H+L) / donkey NGFR 695.15
WM115-B2-rep2
C7
WM-115 Vemurafenib UNC1215 1.0000 0.1067
uM
48
hr
2 1460 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 129.83 NGFR rabbit IgG(H+L) / donkey NGFR 1111.05
WM115-B2-rep2
C8
WM-115 Vemurafenib JW55 1.0000 0.1067
uM
48
hr
2 1482 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 140.32 NGFR rabbit IgG(H+L) / donkey NGFR 1155.40
WM115-B2-rep2
D3
WM-115 Vemurafenib Entinostat 1.0000 0.1067
uM
48
hr
2 1807 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 137.38 NGFR rabbit IgG(H+L) / donkey NGFR 1494.32
WM115-B2-rep2
D4
WM-115 Vemurafenib Azacitidine 1.0000 0.1067
uM
48
hr
2 1410 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 142.24 NGFR rabbit IgG(H+L) / donkey NGFR 1072.40
WM115-B2-rep2
E2
WM-115 Vemurafenib C646 1.0000 0.1067
uM
48
hr
2 1309 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 158.79 NGFR rabbit IgG(H+L) / donkey NGFR 1107.75
WM115-B2-rep2
E3
WM-115 Vemurafenib Tranylcypromine 1.0000 0.1067
uM
48
hr
2 1288 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 136.03 NGFR rabbit IgG(H+L) / donkey NGFR 1117.36
WM115-B2-rep2
G6
WM-115 Vemurafenib UNC0638 1.0000 0.1067
uM
48
hr
2 1283 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 143.28 NGFR rabbit IgG(H+L) / donkey NGFR 1261.16
WM115-B2-rep2
G5