Protein levels measured by imaging in BRAF(V600E/D) melanoma cell lines following treatment with Vemurafenib in combination with chromatin-targeting compounds (immunofluorescence dataset 3 of 4) - Dataset (ID:20276)

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Cell Small Molecule 1 Small Molecule 2 Small Mol 1 Concentration Small Mol 2 Concentration Small Mol Conc Unit Time Point Time Point Unit Replicate Number of Cells Primary Antibody (488) Secondary Antibody (488) Protein Detected (488) Mean Fluorescence Intensity (488) Primary Antibody (647) Secondary Antibody (647) Protein Detected (647) Mean Fluorescence Intensity (647) Plate Name Plate Well
WM-115 Vemurafenib JW55 1.0000 2.6667
uM
48
hr
2 1346 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 130.36 NGFR rabbit IgG(H+L) / donkey NGFR 1010.77
WM115-A2-rep2
D3
WM-115 Vemurafenib PFI-1 1.0000 2.6667
uM
48
hr
2 1357 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 122.24 NGFR rabbit IgG(H+L) / donkey NGFR 628.79
WM115-A2-rep2
B7
WM-115 Vemurafenib UNC669 1.0000 2.6667
uM
48
hr
2 1434 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 128.53 NGFR rabbit IgG(H+L) / donkey NGFR 1073.23
WM115-A2-rep2
B8
WM-115 Vemurafenib Veliparib 1.0000 2.6667
uM
48
hr
2 1323 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 147.36 NGFR rabbit IgG(H+L) / donkey NGFR 1068.09
WM115-A2-rep2
C2
WM-115 Vemurafenib GSK-J1 1.0000 2.6667
uM
48
hr
2 1583 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 129.68 NGFR rabbit IgG(H+L) / donkey NGFR 1085.48
WM115-A2-rep2
B6
WM-115 Vemurafenib Iniparib 1.0000 2.6667
uM
48
hr
2 1379 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 127.25 NGFR rabbit IgG(H+L) / donkey NGFR 992.21
WM115-A2-rep2
B3
WM-115 Vemurafenib CTB 1.0000 2.6667
uM
48
hr
2 1474 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 139.13 NGFR rabbit IgG(H+L) / donkey NGFR 836.64
WM115-A2-rep2
B4
WM-115 Vemurafenib Rocilinostat 1.0000 2.6667
uM
48
hr
2 1454 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 116.84 NGFR rabbit IgG(H+L) / donkey NGFR 520.46
WM115-A2-rep2
B5
WM-115 Vemurafenib Rucaparib 1.0000 2.6667
uM
48
hr
2 1442 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 131.89 NGFR rabbit IgG(H+L) / donkey NGFR 1104.39
WM115-A2-rep2
C3
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1398 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 133.64 NGFR rabbit IgG(H+L) / donkey NGFR 1025.20
WM115-A2-rep2
A7
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1445 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 135.41 NGFR rabbit IgG(H+L) / donkey NGFR 1020.33
WM115-A2-rep2
A8
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1643 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 131.59 NGFR rabbit IgG(H+L) / donkey NGFR 1021.18
WM115-A2-rep2
A9
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1304 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 136.88 NGFR rabbit IgG(H+L) / donkey NGFR 937.20
WM115-A2-rep2
A6
WM-115 Vemurafenib Olaparib 1.0000 2.6667
uM
48
hr
2 1137 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 140.72 NGFR rabbit IgG(H+L) / donkey NGFR 1028.30
WM115-A2-rep2
B2
WM-115 Vemurafenib Belinostat 1.0000 2.6667
uM
48
hr
2 690 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 141.25 NGFR rabbit IgG(H+L) / donkey NGFR 284.20
WM115-A2-rep2
C4
WM-115 Vemurafenib AGK2 1.0000 2.6667
uM
48
hr
2 313 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 133.37 NGFR rabbit IgG(H+L) / donkey NGFR 888.19
WM115-A2-rep2
D5
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1372 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 135.88 NGFR rabbit IgG(H+L) / donkey NGFR 973.52
WM115-A2-rep2
A10
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1297 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 133.03 NGFR rabbit IgG(H+L) / donkey NGFR 965.78
WM115-A2-rep2
A11
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1422 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 173.16 NGFR rabbit IgG(H+L) / donkey NGFR 882.89
WM115-A2-rep2
A2
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1319 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 154.08 NGFR rabbit IgG(H+L) / donkey NGFR 923.84
WM115-A2-rep2
A3
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1454 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 163.37 NGFR rabbit IgG(H+L) / donkey NGFR 947.23
WM115-A2-rep2
A4
WM-115 Vemurafenib 1.0000
uM
48
hr
2 1502 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 143.53 NGFR rabbit IgG(H+L) / donkey NGFR 933.73
WM115-A2-rep2
A5
WM-115 Vemurafenib GSK-J4 1.0000 2.6667
uM
48
hr
2 1545 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 119.21 NGFR rabbit IgG(H+L) / donkey NGFR 1027.05
WM115-A2-rep2
D6
WM-115 Vemurafenib 1.0000
uM
48
hr
2 810 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 133.85 NGFR rabbit IgG(H+L) / donkey NGFR 859.67
WM115-A2-rep2
H7
WM-115 Vemurafenib 1.0000
uM
48
hr
2 845 KI-67 / clone 8D5 mouse IgG(H+L) / donkey KI-67 127.28 NGFR rabbit IgG(H+L) / donkey NGFR 900.40
WM115-A2-rep2
H8