Taselisib KINOMEscan - Dataset (ID:20264)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Taselisib | DRAK1 | 100.0 | 100 | nM |
Taselisib | DRAK1 | 97.0 | 1000 | nM |
Taselisib | DRAK2 | 94.0 | 100 | nM |
Taselisib | DRAK2 | 97.0 | 1000 | nM |
Taselisib | DYRK1A | 83.0 | 100 | nM |
Taselisib | DYRK1A | 99.0 | 1000 | nM |
Taselisib | DYRK1B | 74.0 | 100 | nM |
Taselisib | DYRK1B | 84.0 | 1000 | nM |
Taselisib | DYRK2 | 93.0 | 100 | nM |
Taselisib | DYRK2 | 64.0 | 1000 | nM |
Taselisib | EGFR | 96.0 | 100 | nM |
Taselisib | EGFR | 93.0 | 1000 | nM |
Taselisib | EGFR(E746-A750del) | 89.0 | 100 | nM |
Taselisib | EGFR(E746-A750del) | 97.0 | 1000 | nM |
Taselisib | EGFR(G719C) | 93.0 | 100 | nM |
Taselisib | EGFR(G719C) | 97.0 | 1000 | nM |
Taselisib | EGFR(G719S) | 98.0 | 100 | nM |
Taselisib | EGFR(G719S) | 86.0 | 1000 | nM |
Taselisib | EGFR(L747-E749del, A750P) | 100.0 | 100 | nM |
Taselisib | EGFR(L747-E749del, A750P) | 87.0 | 1000 | nM |
Taselisib | EGFR(L747-S752del, P753S) | 88.0 | 100 | nM |
Taselisib | EGFR(L747-S752del, P753S) | 91.0 | 1000 | nM |
Taselisib | EGFR(L747-T751del,Sins) | 88.0 | 100 | nM |
Taselisib | EGFR(L747-T751del,Sins) | 84.0 | 1000 | nM |
Taselisib | AAK1 | 77.0 | 100 | nM |