Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib DYRK2 93.0 100
nM
Taselisib EGFR 93.0 1000
nM
Taselisib EGFR 96.0 100
nM
Taselisib EGFR(E746-A750del) 97.0 1000
nM
Taselisib EGFR(E746-A750del) 89.0 100
nM
Taselisib EGFR(G719C) 93.0 100
nM
Taselisib EGFR(G719C) 97.0 1000
nM
Taselisib EGFR(G719S) 86.0 1000
nM
Taselisib EGFR(G719S) 98.0 100
nM
Taselisib EGFR(L747-E749del, A750P) 87.0 1000
nM
Taselisib EGFR(L747-E749del, A750P) 100.0 100
nM
Taselisib EGFR(L747-S752del, P753S) 91.0 1000
nM
Taselisib EGFR(L747-S752del, P753S) 88.0 100
nM
Taselisib EGFR(L747-T751del,Sins) 88.0 100
nM
Taselisib EGFR(L747-T751del,Sins) 84.0 1000
nM
Taselisib EGFR(L858R) 99.0 100
nM
Taselisib EGFR(L858R) 90.0 1000
nM
Taselisib EGFR(L858R,T790M) 98.0 1000
nM
Taselisib EGFR(L858R,T790M) 69.0 100
nM
Taselisib EGFR(L861Q) 79.0 1000
nM
Taselisib EGFR(L861Q) 95.0 100
nM
Taselisib EGFR(S752-I759del) 93.0 100
nM
Taselisib EGFR(S752-I759del) 99.0 1000
nM
Taselisib EGFR(T790M) 90.0 100
nM
Taselisib EGFR(T790M) 100.0 1000
nM