Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib FLT3(D835V) 68.0 100
nM
Taselisib EGFR(L858R,T790M) 69.0 100
nM
Taselisib TNK1 69.0 1000
nM
Taselisib MAST1 69.0 1000
nM
Taselisib PAK6 70.0 100
nM
Taselisib HASP 70.0 100
nM
Taselisib MK13 70.0 100
nM
Taselisib CDKL1 71.0 100
nM
Taselisib GRK4 71.0 1000
nM
Taselisib YSK4 71.0 1000
nM
Taselisib RIOK3 71.0 100
nM
Taselisib PAK3 72.0 1000
nM
Taselisib PFCDPK1(P.falciparum) 72.0 1000
nM
Taselisib SRPK3 72.0 100
nM
Taselisib EPHB2 72.0 100
nM
Taselisib M4K1 72.0 1000
nM
Taselisib LRRK2(G2019S) 72.0 100
nM
Taselisib PLK2 73.0 100
nM
Taselisib ERBB4 73.0 1000
nM
Taselisib LTK 73.0 1000
nM
Taselisib CSK 73.0 100
nM
Taselisib RSK2(Kin.Dom.2-C-terminal) 73.0 100
nM
Taselisib RSK3(Kin.Dom.2-C-terminal) 73.0 100
nM
Taselisib ALK(L1196M) 74.0 1000
nM
Taselisib DYRK1B 74.0 100
nM